SCHEMBL7375744

SCHEMBL7375744

NCc1c(O)noc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 6/20 0.42
PTPN1 P18031 1/20 0.41
S1PR1 P21453 1/20 0.38
DPP4 P27487 1/20 0.38
ALDH1A1 P00352 4/20 0.36
IP6K1 Q92551 3/20 0.36
IP6K3 Q96PC2 2/20 0.36
IP6K2 Q9UHH9 2/20 0.36
TP53 P04637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PTGS1 P23219 1/20 0.36
DUSP3 P51452 2/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8376465 0.79 ALDH1A1 (0.37) PTPN1S1PR1ALDH1A1IP6K1IP6K3
SCHEMBL8376467 0.79 ALDH1A1 (0.37) PTPN1S1PR1ALDH1A1IP6K1IP6K3
SCHEMBL7374595 0.78 PTPN1 (0.38) PTPN1ALDH1A1IP6K1IP6K3IP6K2
SCHEMBL8380011 0.78 PTPN1 (0.38) NOTUMPTPN1S1PR1ALDH1A1IP6K1
SCHEMBL8380048 0.78 S1PR1 (0.42) NOTUMPTPN1S1PR1ALDH1A1IP6K1
SCHEMBL8129370 0.77 SLC7A5 (0.46) PTPN1PTGS1
SCHEMBL7159040 0.77 SLC7A5 (0.46) PTPN1PTGS1
SCHEMBL7159035 0.77 SLC7A5 (0.46) PTPN1PTGS1
SCHEMBL8375772 0.76 GCGR (0.45) S1PR1
SCHEMBL8128585 0.75 KIF11 (0.39) PTPN1PTGS1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994107-A1 5-Arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds H. LUNDBECK A/S (DK) 2000-04-19 EP disclosed
EP-0726896-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1996-08-21 EP disclosed
WO-1995012587-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1995-05-11 WO disclosed