SCHEMBL7375868

SCHEMBL7375868

OC(Cc1ccncc1)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.82

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.55
CCR5 P51681 1/20 0.48
CXCR4 P61073 1/20 0.48
TSHR P16473 2/20 0.48
TRPV6 Q9H1D0 1/20 0.48
KDM4E B2RXH2 1/20 0.48
ACHE P22303 1/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380899 0.84 BCHE (0.56) SIGMAR1KDM4EACHE
SCHEMBL5228400 0.80 ACHE (0.60) SIGMAR1CXCR4ACHE
SCHEMBL2953321 0.79 ACHE (0.54) SIGMAR1CXCR4KDM4EACHE
SCHEMBL27691732 0.79 SIGMAR1 (0.48) SIGMAR1TSHRTRPV6KDM4E
SCHEMBL28639634 0.79 ACHE (0.54) SIGMAR1CXCR4KDM4EACHE
SCHEMBL18848489 0.79 ACHE (0.54) SIGMAR1CXCR4KDM4EACHE
SCHEMBL5783247 0.78 CXCR4 (0.46) CXCR4KDM4ECYP3A4CYP2D6
SCHEMBL19450643 0.78 ACHE (0.61) SIGMAR1CXCR4TSHRKDM4EACHE
SCHEMBL1475164 0.77 SIGMAR1 (0.56) SIGMAR1KDM4E
SCHEMBL28565840 0.75 CYP1A2 (0.43) SIGMAR1TSHRKDM4ECYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116846-A N-ARALKYL PIPERIDINE DERIVATIVES AS PSYCHOTROPIC DRUGS DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-05-26 US disclosed
EP-0449186-A2 N-aralkyl piperidine derivatives as psychotropic drugs THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-10-02 EP disclosed