SCHEMBL7377018

SCHEMBL7377018

CCC(Cl)N1CCC(NC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.59
SLC6A12 P48065 1/20 0.59
TMEM97 Q5BJF2 1/20 0.59
SIGMAR1 Q99720 1/20 0.59
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
KMT2A Q03164 6/20 0.55
CTSB P07858 1/20 0.52
CTSS P25774 1/20 0.52
CTSK P43235 1/20 0.52
CTSC P53634 1/20 0.52
TSHR P16473 2/20 0.52
USP2 O75604 1/20 0.52
CCR3 P51677 1/20 0.52
MEN1 O00255 3/20 0.51
DRD2 P14416 1/20 0.51
DRD4 P21917 1/20 0.51
HTR1A P08908 1/20 0.51
HTR7 P34969 1/20 0.51
HRH3 Q9Y5N1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7389264 0.88 NPSR1 (0.58) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL20147581 0.84 HRH3 (0.68) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL21652025 0.81 MCHR1 (0.68) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL4749226 0.79 NPC1 (0.67) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL14021836 0.79 NPC1 (0.67) MCHR1SLC6A12TMEM97SIGMAR1NPC1
Fk-962 SCHEMBL239762 0.77 KMT2A (0.69) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL532160 0.77 RAB9A (0.83) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL14679122 0.76 NPC1 (0.58) NPC1RAB9AKMT2ATSHRMEN1
SCHEMBL6379927 0.76 MCHR1 (0.69) MCHR1SLC6A12TMEM97SIGMAR1NPC1
SCHEMBL14004335 0.76 NPC1 (0.61) MCHR1SLC6A12TMEM97SIGMAR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012147-A2 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-28 EP disclosed
WO-1999006387-A2 O-SUBSTITUTED HYDROXYCUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1999-02-11 WO disclosed