Fk-962

Fk-962

SCHEMBL239762

CC(=O)N1CCC(NC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.69
USP2 O75604 1/20 0.64
TSHR P16473 1/20 0.64
NPC1 O15118 1/20 0.63
RAB9A P51151 1/20 0.63
MEN1 O00255 4/20 0.62
POLB P06746 2/20 0.59
SLC6A12 P48065 1/20 0.59
TMEM97 Q5BJF2 1/20 0.59
MCHR1 Q99705 1/20 0.59
SIGMAR1 Q99720 1/20 0.59
CRBN Q96SW2 1/20 0.58
CTSB P07858 1/20 0.58
CTSS P25774 1/20 0.58
CTSK P43235 1/20 0.58
CTSC P53634 1/20 0.58
HDAC4 P56524 1/20 0.58
CCR3 P51677 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19480105 0.87 NPC1 (0.65) KMT2AUSP2TSHRNPC1RAB9A
SCHEMBL1424917 0.86 KMT2A (0.66) KMT2AUSP2TSHRNPC1RAB9A
SCHEMBL14590545 0.85 NPSR1 (0.67) KMT2ANPC1RAB9AMEN1POLB
SCHEMBL4749226 0.85 NPC1 (0.67) KMT2AUSP2TSHRNPC1RAB9A
SCHEMBL1425012 0.85 KMT2A (0.64) KMT2AUSP2TSHRNPC1RAB9A
SCHEMBL6539130 0.84 KMT2A (0.67) KMT2AUSP2TSHRNPC1RAB9A
SCHEMBL19356248 0.83 CRBN (0.56) KMT2ATSHRMEN1CRBNHDAC4
SCHEMBL17572986 0.83 KMT2A (0.63) KMT2ATSHRMEN1POLBCRBN
SCHEMBL14797275 0.82 CRBN (0.55) KMT2ATSHRMEN1POLBCRBN
SCHEMBL532160 0.82 RAB9A (0.83) KMT2AUSP2TSHRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 125 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2157082-B1 NEURITE FORMATION PROMOTER SENJU PHARMA CO (JP) 2016-06-08 EP claimed
US-8637544-B2 Neurite formation promoter SENJU PHARMACEUTICAL CO., LTD. (JP) 2014-01-28 US claimed
EP-1140836-B1 AMIDE COMPOUNDS ASTELLAS PHARMA INC (JP) 2011-03-23 EP claimed
US-20100144792-A1 NEURITE FORMATION PROMOTER SENJU PHARMACEUTICAL CO., LTD. (JP) 2010-06-10 US claimed
CN-101687795-A Neuritogenesis promoter SENJU PHARMA CO 2010-03-31 CN claimed
EP-2157082-A1 NEURITE FORMATION PROMOTER Senju Pharmaceutical Co., Ltd. (JP) 2010-02-24 EP claimed
US-6710043-B1 POSSESS THE POTENTIATION OF THE CHOLINERGIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-03-23 US claimed
US-12637455-B2 Naphthyridine and pyrido[3,4-c]pyridazine derivatives as GABAA α5 receptor modulators RICHTER GEDEON NYRT. (HU) 2026-05-26 US disclosed
EP-4126858-B1 DIHYDRO-2-PYRROLO[3,4-C]PYRIDINE DERIVATIVES AS GABAA A5 RECEPTOR MODULATORS RICHTER GEDEON NYRT (HU) 2026-03-18 EP disclosed
US-12534458-B2 Spiropiperidine allosteric modulators of nicotinic acetylcholine receptors MERCK SHARP & DOHME LLC (US) 2026-01-27 US disclosed
EP-3856342-B1 BICYCLIC DERIVATIVES AS GABAA A5 RECEPTOR MODULATORS RICHTER GEDEON NYRT (HU) 2025-12-10 EP disclosed
US-20250344963-A1 METHODS FOR ACQUIRING AND ANALYZING NEUROMELANIN-SENSITIVE MRI UNIV OF OTTAWA INSTITUTE OF MENTAL HEALTH RESEARCH (CA) 2025-11-13 US disclosed
US-20250302913-A1 LACRIPEP PROMOTES NEUROREGENERATION AND MAINTAINS EPITHELIAL PROGENITOR CELL IDENTITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-10-02 US disclosed
WO-2002020016-A1 AGENT FOR MODULATING EXCITATORY SYNAPTIC TRANSMISSION COMPRISING A COMPOUND HAVING ALPHA α7 NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO, LTD (JP) 2002-03-14 WO disclosed
CN-1336917-A Amide compounds FUJISAWA PHARMACEUTICAL CO (JP) 2002-02-20 CN disclosed
US-6344358-B1 ADMINISTERING SOMATOSTATIN RELEASING AGENT TO TREAT BRAIN, PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS SUCH AS SCHIZOPHRENIA, AMNESIA, BIPOLAR DISORDER, ALZHEIMER*S DISEASE AND PARKINSON*S DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-05 US disclosed
WO-2000072834-A9 AGENT FOR EXPRESSION OF LONG-TERM POTENTIATION OF SYNAPTIC TRANSMISSION COMPRISING COMPOUND HAVING BRAIN SOMATOSTATIN ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO (JP) 2001-12-20 WO disclosed
EP-1140836-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-10 EP disclosed
WO-2000072834-A2 AGENT FOR EXPRESSION OF LONG-TERM POTENTIATION OF SYNAPTIC TRANSMISSION COMPRISING COMPOUND HAVING BRAIN SOMATOSTATIN ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-12-07 WO disclosed
WO-2000042011-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12534458-B2 Spiropiperidine allosteric modulators of nicotinic acetylcholine receptors CHRNA6, CHRNA7, CHRNA5 KMT2A 3415/4885USP2 3853/4885TSHR 216/4885
US-12637455-B2 Naphthyridine and pyrido[3,4-c]pyridazine derivatives as GABAA α5 receptor modulators GABRA5, GABRA1, GABRB1 KMT2A 4249/4885USP2 4371/4885TSHR 263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.