SCHEMBL7377241

SCHEMBL7377241

[CH2]C(CC(N)=O)c1cc(N)cc([N+](=O)[O-])c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 5/20 0.38
ALDH1A1 P00352 5/20 0.38
LMNA P02545 2/20 0.38
GRM8 O00222 1/20 0.38
GRM4 Q14833 1/20 0.38
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GPR35 Q9HC97 1/20 0.34
TSHR P16473 3/20 0.33
MITF O75030 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7373745 0.81 VCAM1 (0.51) SMN1; SMN2CYP3A4MAPTALDH1A1GRM8
Urea SCHEMBL3678424 0.73 SMN1; SMN2 (0.63) NPC1SMN1; SMN2CYP3A4MAPTALDH1A1
SCHEMBL7379785 0.72 TNF (0.40) GRM4
SCHEMBL7080519 0.71 NPC1 (0.46) NPC1SMN1; SMN2CYP3A4MAPTALDH1A1
SCHEMBL13458416 0.71 ALDH1A1 (0.47) NPC1CYP3A4MAPTALDH1A1LMNA
SCHEMBL7379834 0.71 CYP2C19 (0.37) CYP3A4ALDH1A1HTTTSHR
Acrylamide SCHEMBL27801304 0.69 SMN1; SMN2 (0.53) NPC1SMN1; SMN2CYP3A4MAPTALDH1A1
SCHEMBL8417924 0.69 SMN1; SMN2 (0.44) NPC1SMN1; SMN2CYP3A4MAPTALDH1A1
SCHEMBL6664755 0.69 GPR35 (0.41) NPC1SMN1; SMN2CYP3A4MAPTALDH1A1
SCHEMBL539064 0.69 ALDH1A1 (0.60) NPC1SMN1; SMN2CYP3A4MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed