SCHEMBL7377281

SCHEMBL7377281

CCOC(=O)C1=C(C)N2OCCOC2=C(C(=O)OCC)C1(C)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1D Q01668 4/20 0.38
CACNA1C Q13936 3/20 0.38
CACNA1F O60840 2/20 0.38
CACNA1S Q13698 2/20 0.38
ALDH1A1 P00352 4/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 3/20 0.36
MAPT P10636 4/20 0.36
ADORA3 P0DMS8 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
THRB P10828 1/20 0.34
POLB P06746 1/20 0.34
RECQL P46063 1/20 0.34
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2907995 0.70 ALDH1A1 (0.44) CACNA1DCACNA1CCACNA1FCACNA1SALDH1A1
SCHEMBL4880017 0.64 TSHR (0.38) ALDH1A1GAASMN1; SMN2KDM4EMAPT
SCHEMBL7382729 0.63 TSHR (0.37) ALDH1A1GAAKDM4EMAPTL3MBTL1
SCHEMBL5445916 0.63 CACNA1D (0.42) CACNA1DCACNA1CCACNA1FCACNA1SALDH1A1
SCHEMBL1523174 0.63 ALDH1A1 (0.67) ALDH1A1GAASMN1; SMN2MAPTL3MBTL1
SCHEMBL4755372 0.60 TSHR (0.39) ALDH1A1GAASMN1; SMN2KDM4EMAPT
SCHEMBL6737967 0.60 OPRM1 (0.61) CACNA1DCACNA1CCACNA1FCACNA1SALDH1A1
SCHEMBL7383668 0.60 CACNA1C (0.47) CACNA1DCACNA1CCACNA1FCACNA1SALDH1A1
SCHEMBL8664750 0.60 ALDH1A1 (0.53) CACNA1DALDH1A1GAASMN1; SMN2KDM4E
Ethyl Acetate SCHEMBL27861469 0.60 RAB9A (0.52) ALDH1A1GAASMN1; SMN2KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4525478-A Certain 4-aryl-1,4-dihydro-3,5-pyridinedicarboxylates having vasodilating and anti-hypertensive properties FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1985-06-25 US disclosed
US-4370334-A VASODILATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-01-25 US disclosed
US-4338322-A 1,4-Dihydropyridine derivatives, pharmaceutical compositions containing same and methods of effecting vasodilation using same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1982-07-06 US disclosed
US-4284634-A HYPOTENSIVE VASODILATORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-08-18 US disclosed
US-4145432-A 6-ACYLORYALKYL-1,4-DIHYDROPYRIDINE DERIVATIVES AND A METHOD OF EFFECTING VASODILATION THEREWITH FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1979-03-20 US disclosed