SCHEMBL7377758

SCHEMBL7377758

CC(C)c1c(CO)[nH]c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.49
CDK1 P06493 1/20 0.49
CCNB1 P14635 1/20 0.49
CCNB3 Q8WWL7 1/20 0.49
KIF11 P52732 3/20 0.46
ALDH1A1 P00352 5/20 0.45
HSD17B10 Q99714 2/20 0.45
GPR3 P46089 1/20 0.45
VDR P11473 1/20 0.44
SIRT1 Q96EB6 2/20 0.41
HTT P42858 2/20 0.41
TSHR P16473 1/20 0.41
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
AURKA O14965 1/20 0.40
MAPK10 P53779 1/20 0.40
RIPK1 Q13546 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14365065 0.84 CCNB2 (0.50) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL29443497 0.82 KIF11 (0.46) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL9457713 0.80 KDM4E (0.53) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL8247023 0.79 CCNB2 (0.46) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL23429368 0.76 CCNB2 (0.53) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL13301938 0.76 AHR (0.55) KIF11ALDH1A1HSD17B10GPR3HTT
SCHEMBL10280325 0.75 CCNB2 (0.56) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL30234429 0.75 CCNB2 (0.56) CCNB2CDK1CCNB1CCNB3KIF11
SCHEMBL7373159 0.74 DRD2 (0.52) KIF11ALDH1A1HSD17B10GPR3HTT
SCHEMBL8997990 0.73 VDR (0.67) CCNB2CDK1CCNB1CCNB3KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420086-B1 Pyrimidoindole derivatives and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO (JP) 1995-12-13 EP disclosed
US-5256780-A Serotonin antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-10-26 US disclosed
US-5180728-A Antagonists of 5-hydroxytryptamine FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1993-01-19 US disclosed
EP-0420086-A2 Pyrimidoindole derivatives and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-04-03 EP disclosed