SCHEMBL7378397

SCHEMBL7378397

Fc1ccn2c(Cc3ncc[nH]3)c(-c3ccc(Cl)cc3)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 1/20 0.39
KDM4E B2RXH2 4/20 0.38
POLB P06746 2/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NAMPT P43490 2/20 0.38
KCNK3 O14649 3/20 0.37
KCNK9 Q9NPC2 3/20 0.37
SLC2A1 P11166 2/20 0.37
ALDH1A1 P00352 2/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
GAA P10253 1/20 0.35
SLC2A3 P11169 1/20 0.35
SLC2A4 P14672 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7407222 0.90 KDM4E (0.40) KDM4EPOLBNPC1HTTRAB9A
SCHEMBL7372340 0.89 SIRT5 (0.41) SIRT5POLBNAMPTALDH1A1
SCHEMBL7377978 0.86 KCNK3 (0.40) KDM4EPOLBNPC1HTTRAB9A
SCHEMBL7379148 0.83 PSMD14 (0.40) KDM4EPOLBNPC1HTTRAB9A
SCHEMBL7237846 0.78 MAPK13 (0.36) SIRT5KDM4EPOLBNPC1HTT
SCHEMBL7412126 0.77 DPP4 (0.39) POLBNAMPTSLC2A1GAATAAR1
SCHEMBL7554629 0.75 KCNK3 (0.47) KCNK3KCNK9
SCHEMBL7410232 0.74 NR1H4 (0.39) KDM4EPOLBNPC1HTTRAB9A
SCHEMBL22627384 0.71 CYP11B1 (0.64) KDM4EPOLBNPC1HTTRAB9A
SCHEMBL22615010 0.71 CYP11B1 (0.44) KDM4EPOLBNPC1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002002557-A2 2-PHENYLIMIDAZO[1,2-A]PYRIDINE DERIVATIVES: A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-01-10 WO disclosed