SCHEMBL7378673

SCHEMBL7378673

CC(C)(C)OC(=O)CNc1ccc(OCc2ccccc2)cc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 4/20 0.49
CTSL P07711 4/20 0.49
MAOB P27338 1/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 2/20 0.46
PKM P14618 1/20 0.46
MCL1 Q07820 2/20 0.44
BCL2A1 Q16548 1/20 0.43
NR4A2 P43354 2/20 0.43
SLC16A3 O15427 1/20 0.43
NR4A1 P22736 1/20 0.43
NR4A3 Q92570 1/20 0.43
HPGD P15428 1/20 0.42
MDH2 P40926 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
LTA4H P09960 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15589680 0.89 MAOB (0.43) CTSVCTSLMAOBALDH1A1KDM4E
SCHEMBL19159330 0.89 SIRT2 (0.44) CTSVCTSLMAOBKDM4ESIRT2
SCHEMBL7381558 0.85 CTSV (0.52) CTSVCTSLMAOBALDH1A1KDM4E
SCHEMBL19160125 0.82 LTA4H (0.46) MAOBKDM4ESMN1; SMN2LTA4HMEN1
SCHEMBL7374213 0.80 MAPT (0.45) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL28302706 0.80 PDK1 (0.57) CTSVCTSLMAOBALDH1A1KDM4E
SCHEMBL5956241 0.79 KDM4E (0.56) ALDH1A1KDM4EHPGDSMN1; SMN2MEN1
SCHEMBL22762667 0.78 KDM4E (0.60) CTSVCTSLMAOBALDH1A1KDM4E
SCHEMBL646567 0.77 BRD4 (0.42)
SCHEMBL3916435 0.77 LTA4H (0.39) LTA4HMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171166-A1 BENZODIAZEPINE DERIVATIVES FOR IMAGING THROMBI Diatide, Inc. (US) 2002-01-16 EP disclosed
US-6171578-B1 GLYCOPROTEIN IIB/IIIA RECEPTOR-BINDING BENZODIAZEPINE DERIVATIVES COVALENTLY LINKED TO METAL ION CHELATORS. DIATIDE, INC. 2001-01-09 US disclosed
WO-2000061195-A1 BENZODIAZEPINE DERIVATIVES FOR IMAGING THROMBI DIATIDE, INC. (US) 2000-10-19 WO disclosed