SCHEMBL7379162

SCHEMBL7379162

CCOC(=O)CCCCCOc1ccccc1NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
EBP Q15125 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP2C19 P33261 1/20 0.43
PPARG P37231 1/20 0.42
PTPN1 P18031 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
EPHX2 P34913 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16010936 0.85 NLRP3 (0.45) GAAALDH1A1TSHR
SCHEMBL18078943 0.83 KMT2A (0.60) GAAEBPSIGMAR1KMT2AALDH1A1
SCHEMBL7369166 0.82 LTA4H (0.48) GAAKMT2AALDH1A1PPARGTDP1
SCHEMBL14363211 0.81 MAPT (0.52) GAAKMT2AALDH1A1CYP2C19TDP1
SCHEMBL29991286 0.81 GAA (0.63) GAAKMT2AALDH1A1CYP2C19TDP1
SCHEMBL5655945 0.81 GAA (0.63) GAAKMT2AALDH1A1CYP2C19TDP1
SCHEMBL28125405 0.79 LMNA (0.52) GAAEBPSIGMAR1KMT2AALDH1A1
SCHEMBL8159189 0.79 GAA (0.58) GAAKMT2AALDH1A1CYP2C19PPARG
SCHEMBL14363180 0.79 HDAC8 (0.53) ALDH1A1
SCHEMBL8162740 0.78 GAA (0.56) GAAKMT2AALDH1A1CYP2C19TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed