SCHEMBL7380141

SCHEMBL7380141

[CH2]c1cccc(-n2ncc(N)n2)c1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.34
GRM5 P41594 1/20 0.34
MEN1 O00255 2/20 0.32
NPC1 O15118 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
RAB9A P51151 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KDM4E B2RXH2 1/20 0.31
STAT1 P42224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372783 0.79 P2RX7 (0.34) P2RX7GRM5MEN1NPC1ALDH1A1
SCHEMBL18039129 0.77 P2RX7 (0.53) P2RX7MEN1NPC1ALDH1A1MAPT
SCHEMBL7374338 0.76 ADORA2A (0.39) P2RX7GRM5MEN1NPC1ALDH1A1
SCHEMBL10965939 0.76 P2RX7 (0.45) P2RX7
SCHEMBL7370991 0.76 LSS (0.32) P2RX7GRM5
SCHEMBL7377818 0.76 P2RX7 (0.45) P2RX7GRM5
SCHEMBL7376072 0.74 ACLY (0.35) MEN1NPC1ALDH1A1MAPTRAB9A
SCHEMBL7381168 0.72 ADORA2A (0.37) P2RX7GRM5
SCHEMBL7380060 0.72 P2RX7 (0.33) P2RX7GRM5KMT2A
SCHEMBL10783183 0.70 TP53 (0.51) GRM5NPC1ALDH1A1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO claimed
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO disclosed