SCHEMBL7380729

SCHEMBL7380729

O=C(O)C(CCc1ccccc1)NCC(C(=O)O)C1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACE P12821 9/20 0.49
TAAR1 Q96RJ0 1/20 0.47
EPHX2 P34913 4/20 0.45
MME P08473 1/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
EPHX1 P07099 1/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7382520 0.95 MME (0.47) ACEMME
SCHEMBL5652285 0.84 L3MBTL1 (0.52) TAAR1EPHX2HTTL3MBTL1NPC1
SCHEMBL7539729 0.79 EPHX2 (0.54) TAAR1EPHX2HTTL3MBTL1NPC1
Cyclohexylglycyl SCHEMBL7423505 0.77 ACE (0.46) ACETAAR1EPHX2NPC1TP53
SCHEMBL27495306 0.75 CYP2C9 (0.61) ACETAAR1EPHX2MMEEPHX1
SCHEMBL7428877 0.75 TAAR1 (0.52) ACETAAR1EPHX2NPC1TP53
SCHEMBL8249114 0.75 MME (0.56) ACEEPHX2MME
SCHEMBL5869478 0.75 MME (0.56) ACEEPHX2MME
SCHEMBL10482542 0.74 MME (0.56) ACEMMEEPHX1TSHRSMN1; SMN2
SCHEMBL10482537 0.74 MME (0.56) ACEMMEEPHX1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000066104-A9 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARM INC (US) 2002-08-29 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed
EP-1183019-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF Millennium Pharmaceuticals, Inc. (US) 2002-03-06 EP disclosed
WO-2000066104-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2000-11-09 WO disclosed