Cladrin

Cladrin

SCHEMBL738092

COc1ccc(-c2coc3cc(O)ccc3c2=O)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 1.00
HSD17B10 Q99714 9/20 1.00
MAPT P10636 6/20 1.00
NPC1 O15118 6/20 1.00
RAB9A P51151 6/20 1.00
TP53 P04637 3/20 1.00
MAPK1 P28482 1/20 1.00
POLB P06746 2/20 0.84
HMGB1 P09429 1/20 0.84
ALDH1A1 P00352 9/20 0.73
HPGD P15428 8/20 0.73
SMN1; SMN2 Q16637 5/20 0.73
CYP3A4 P08684 4/20 0.73
HDAC6 Q9UBN7 3/20 0.73
CYP2D6 P10635 2/20 0.73
CYP2C9 P11712 2/20 0.73
MAOA P21397 2/20 0.73
MAOB P27338 2/20 0.73
CYP2C19 P33261 2/20 0.73
MEN1 O00255 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Calycosin SCHEMBL30335127 0.91 KDM4E (1.00) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL2069826 0.91 KDM4E (0.84) KDM4EHSD17B10MAPTNPC1RAB9A
Calycosin SCHEMBL73013 0.91 KDM4E (1.00) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL29788255 0.91 KDM4E (0.84) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL30238115 0.91 KDM4E (0.83) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL28124530 0.89 KDM4E (0.80) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL13904731 0.87 KDM4E (0.77) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL12206681 0.87 KDM4E (0.77) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL10560560 0.86 PTPN1 (0.77) KDM4EHSD17B10MAPTNPC1RAB9A
SCHEMBL13631294 0.86 MAPT (0.77) KDM4EHSD17B10MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9408826-B2 Isoflavone anti-viral compounds Kineta, Inc. (US) 2016-08-09 US disclosed
US-9408826-B2 Isoflavone anti-viral compounds Kineta, Inc. (US) 2016-08-09 US disclosed
US-9408826-B2 Isoflavone anti-viral compounds Kineta, Inc. (US) 2016-08-09 US disclosed
EP-2560652-A2 ANTI-VIRAL COMPOUNDS Kineta, Inc. (US) 2013-02-27 EP disclosed
US-8138184-B2 Isoxazole derivatives and pharmaceutical compositions comprising the same KAOHSIUNG MEDICAL UNIVERSITY (TW) 2012-03-20 US disclosed
US-20110262482-A1 ANTI-VIRAL COMPOUNDS Kineta, Inc. (US) 2011-10-27 US disclosed
US-20110262482-A1 ANTI-VIRAL COMPOUNDS Kineta, Inc. (US) 2011-10-27 US disclosed
US-20110262482-A1 ANTI-VIRAL COMPOUNDS Kineta, Inc. (US) 2011-10-27 US disclosed
WO-2011133728-A2 ANTI-VIRAL COMPOUNDS Kineta, Inc. (US) 2011-10-27 WO disclosed
WO-2011133728-A2 ANTI-VIRAL COMPOUNDS Kineta, Inc. (US) 2011-10-27 WO disclosed
US-7247734-B2 3,4-diarylpyrazoles and their use in the therapy of cancer VERNALIS (CAMBRIDGE) LIMITED (GB) 2007-07-24 US disclosed
WO-2006099681-A1 ISOFLAVONOID DIMERS NOVOGEN RESEARCH PTY LTD (AU) 2006-09-28 WO disclosed
US-20050222230-A1 3,4-diarylpyrazoles and their use in the therapy of cancer VERNALIS (CAMBRIDGE) LIMITED (GB) 2005-10-06 US disclosed
EP-1456180-A1 3,4-DIARYLPYRAZOLES AND THEIR USE IN THE THERAPY OF CANCER Vernalis (Oxford) Ltd (GB) 2004-09-15 EP disclosed
WO-2003055860-A1 3,4-DIARYLPYRAZOLES AND THEIR USE IN THE THERAPY OF CANCER VERNALIS (CAMBRIDGE) LIMITED (GB) 2003-07-10 WO disclosed
EP-0710234-A1 ISOFLAVONE DERIVATIVES CHINOIN LTD. (HU) 1996-05-08 EP disclosed
WO-1995003293-A1 ISOFLAVONE DERIVATIVES CHINOIN LTD. (HU) 1995-02-02 WO disclosed
EP-0478558-B1 AN IMPROVED PROCESS FOR THE PREPARATION OF SUBSTITUTED ISOFLAVONE DERIVATIVES CHINOIN GYOGYSZER ES VEGYESZET (HU) 1994-02-02 EP disclosed
US-5247102-A Cyclization of a resorcinol derivative with ethyl orthoformate in the presence of a base CHINOIN GYOGYSZER- ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1993-09-21 US disclosed
WO-1991015483-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF SUBSTITUTED ISOFLAVONE DERIVATIVES CHINOIN GYÓGYSZER ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT (HU) 1991-10-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110262482-A1 ANTI-VIRAL COMPOUNDS MAVS, EIF2AK2, IRF3 KDM4E 2601/4885HSD17B10 4165/4885MAPT 3520/4885
US-20050222230-A1 3,4-diarylpyrazoles and their use in the therapy of cancer HSP90AB1, HSP90AA1, HSP90AB2P KDM4E 1999/4885HSD17B10 222/4885MAPT 4683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.