SCHEMBL7382010

SCHEMBL7382010

[CH2]c1cccc(C(=O)Nc2ncc(CC)s2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
TSHR P16473 1/20 0.53
CCNE1 P24864 2/20 0.52
CDK2 P24941 2/20 0.52
CDK5 Q00535 2/20 0.52
RAB9A P51151 4/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 3/20 0.48
NPC1 O15118 3/20 0.48
THRB P10828 1/20 0.48
MAPK9 P45984 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KDR P35968 1/20 0.48
SCD O00767 4/20 0.48
KDM4E B2RXH2 3/20 0.46
HPGD P15428 3/20 0.46
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8594861 0.86 ALDH1A1 (0.57) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL11919154 0.84 ALDH1A1 (0.70) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL7352140 0.83 SMN1; SMN2 (0.60) ALDH1A1RAB9AMEN1KMT2AMAPT
SCHEMBL7372009 0.83 RAB9A (0.46) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL7379218 0.81 NPC1 (0.49) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL7379033 0.81 KDR (0.51) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL7381091 0.77 HSD17B1 (0.44) ALDH1A1RAB9AMEN1KMT2AMAPT
SCHEMBL4756006 0.75 SCD (0.51) ALDH1A1TSHRCCNE1CDK2CDK5
SCHEMBL7375409 0.75 MAPK1 (0.54) ALDH1A1TSHRRAB9AMAPTNPC1
SCHEMBL7348805 0.74 MEN1 (0.71) ALDH1A1TSHRRAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO claimed
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP disclosed
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO disclosed