SCHEMBL7384168

SCHEMBL7384168

COc1cc2c(cc1OC)C(C#Cc1ccccn1)=CCC2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.43
CYP1A2 P05177 2/20 0.43
PDE10A Q9Y233 1/20 0.42
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HCRTR1 O43613 1/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
MAOA P21397 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
PDE4A P27815 1/20 0.38
GPR84 Q9NQS5 1/20 0.38
PKM P14618 1/20 0.38
RAD52 P43351 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431944 0.79 GRM5 (0.51) GRM5CYP1A2
Hydrochloric Acid SCHEMBL7377474 0.78 GRM5 (0.50) GRM5CYP1A2
SCHEMBL1669168 0.71 KDM4E (0.46) CYP1A2KDM4EALDH1A1GAAMAPT
SCHEMBL28209834 0.66 PDE10A (0.47) PDE10AKDM4EALDH1A1GAAMAPT
SCHEMBL4980429 0.65 GRM5 (0.68) GRM5NPC1RAB9AHCRTR1
Methyl Alcohol SCHEMBL28902013 0.65 GRM5 (0.67) GRM5CYP1A2ALDH1A1MAPTPKM
SCHEMBL352291 0.64 GRM5 (0.65) GRM5CYP1A2TDP1
SCHEMBL21360714 0.64 MAOA (0.56) CYP1A2KDM4EALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL3839867 0.64 GRM5 (0.67) GRM5NPC1RAB9AHCRTR1TDP1
SCHEMBL8887830 0.63 ALDH1A1 (0.50) GRM5CYP1A2NPC1RAB9AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed