SCHEMBL7384642

SCHEMBL7384642

CCCOC(=O)C1=C(C)NC(C)=C(S(=O)(=O)c2ccc(O)cc2)C1c1cccc(Cl)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.56
KDM4E B2RXH2 3/20 0.56
CYP3A4 P08684 3/20 0.56
ABCB11 O95342 3/20 0.56
TBXA2R P21731 3/20 0.56
ADRA1A P35348 3/20 0.56
SLC6A3 Q01959 3/20 0.56
MEN1 O00255 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C19 P33261 2/20 0.56
KMT2A Q03164 2/20 0.56
HIF1A Q16665 2/20 0.56
HSD17B10 Q99714 2/20 0.56
ALDH1A1 P00352 2/20 0.56
TSHR P16473 2/20 0.56
ABCB1 P08183 2/20 0.56
ADORA3 P0DMS8 2/20 0.56
ADRB3 P13945 2/20 0.56
OPRK1 P41145 2/20 0.56
SCN5A Q14524 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7385058 0.95 ALDH1A1 (0.54) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7376680 0.93 TBXA2R (0.48) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7381502 0.93 CYP2C9 (0.64) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7376670 0.88 ALDH1A1 (0.51) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7376040 0.88 KDM4E (0.61) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7385349 0.86 KDM4E (0.54) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL9765752 0.86 CYP3A4 (0.51) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7385182 0.85 CYP2C9 (0.49) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7383535 0.85 CYP2C9 (0.48) CYP2C9KDM4ECYP3A4ABCB11TBXA2R
SCHEMBL7381800 0.85 CYP2C9 (0.48) CYP2C9KDM4ECYP3A4ABCB11TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4889866-A CARDIOVASCULAR DISEASES, HYPOTENSIVE AGENTS, CONGESTIVE HEART FAILURE SYNTEX (U.S.A.) INC. (US) 1989-12-26 US disclosed