SCHEMBL7385349

SCHEMBL7385349

CCOC(=O)C1=C(C)NC(C)=C(S(=O)(=O)c2ccc(O)cc2)C1c1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
TSHR P16473 3/20 0.54
ALDH1A1 P00352 3/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CYP2C9 P11712 3/20 0.53
TBXA2R P21731 3/20 0.53
ADRA1A P35348 3/20 0.53
SLC6A3 Q01959 3/20 0.53
CYP3A4 P08684 3/20 0.53
HSD17B10 Q99714 3/20 0.53
ADORA3 P0DMS8 3/20 0.53
ABCB11 O95342 3/20 0.53
LMNA P02545 3/20 0.53
MEN1 O00255 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2C19 P33261 2/20 0.53
KMT2A Q03164 2/20 0.53
HIF1A Q16665 2/20 0.53
ABCB1 P08183 2/20 0.53
ADRB3 P13945 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381502 0.93 CYP2C9 (0.64) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL7376680 0.93 TBXA2R (0.48) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL7376670 0.91 ALDH1A1 (0.51) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL7382103 0.90 KDM4E (0.56) KDM4ETSHRALDH1A1CYP2C9TBXA2R
SCHEMBL7377019 0.89 KDM4E (0.50) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL7384908 0.87 CYP2C9 (0.43) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL7382382 0.87 NR3C2 (0.45) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL7385356 0.87 ALOX15 (0.52) KDM4ECYP2C9TBXA2RSLC6A3CYP3A4
SCHEMBL7384642 0.86 CYP2C9 (0.56) KDM4ETSHRALDH1A1SMN1; SMN2CYP2C9
SCHEMBL9765752 0.85 CYP3A4 (0.51) KDM4ETSHRALDH1A1CYP2C9TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4889866-A CARDIOVASCULAR DISEASES, HYPOTENSIVE AGENTS, CONGESTIVE HEART FAILURE SYNTEX (U.S.A.) INC. (US) 1989-12-26 US disclosed