SCHEMBL9765752

SCHEMBL9765752

CCCOC(=O)C1=C(C)NC(C)=C(S(=O)(=O)c2ccccc2)C1c1ccccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.51
NR1I2 O75469 2/20 0.51
LMNA P02545 4/20 0.48
CYP2C9 P11712 3/20 0.48
TBXA2R P21731 3/20 0.48
ADRA1A P35348 3/20 0.48
SLC6A3 Q01959 3/20 0.48
ABCB11 O95342 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
MEN1 O00255 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 2/20 0.48
HIF1A Q16665 2/20 0.48
HSD17B10 Q99714 2/20 0.48
ABCB1 P08183 2/20 0.48
ADORA3 P0DMS8 2/20 0.48
ADRB3 P13945 2/20 0.48
OPRK1 P41145 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7376680 0.93 TBXA2R (0.48) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7381554 0.91 KDM4E (0.47) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7376670 0.87 ALDH1A1 (0.51) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7384642 0.86 CYP2C9 (0.56) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7376239 0.86 ALDH1A1 (0.50) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7384442 0.86 KDM4E (0.53) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL11367250 0.86 CYP3A4 (0.42) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7385349 0.85 KDM4E (0.54) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7382103 0.84 KDM4E (0.56) CYP3A4NR1I2LMNACYP2C9TBXA2R
SCHEMBL7379245 0.83 CYP2C9 (0.49) CYP3A4NR1I2LMNACYP2C9TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed