SCHEMBL7385065

SCHEMBL7385065

CCOC(=O)[C@H](Cc1c[nH]c2cc(OC)ccc12)NC=O

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
MAPT P10636 6/20 0.50
TP53 P04637 2/20 0.50
LMNA P02545 1/20 0.50
THRB P10828 1/20 0.50
SCN9A Q15858 1/20 0.50
HTR2A P28223 1/20 0.46
TACR1 P25103 1/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ITGB2 P05107 1/20 0.46
ICAM1 P05362 1/20 0.46
ITGAL P20701 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7385062 1.00 MTNR1A (0.51) MTNR1AMTNR1BMAPTTP53LMNA
SCHEMBL29421743 0.82 APLNR (0.47) MAPTMEN1KMT2AALDH1A1
SCHEMBL6301729 0.81 SCN9A (0.60) MTNR1AMTNR1BMAPTSCN9AHTR2A
SCHEMBL30663629 0.81 SCN9A (0.60) MTNR1AMTNR1BMAPTSCN9AHTR2A
SCHEMBL21384322 0.81 SCN9A (0.60) MTNR1AMTNR1BMAPTSCN9AHTR2A
SCHEMBL19392083 0.76 KMT2A (0.64) MAPTTP53MEN1KMT2A
SCHEMBL16645246 0.76 MTNR1A (0.58) MTNR1AMTNR1BMAPTSCN9AHTR2A
SCHEMBL17938401 0.76 MTNR1A (0.58) MTNR1AMTNR1BMAPTSCN9AHTR2A
SCHEMBL8490235 0.76 KMT2A (0.64) MAPTTP53MEN1KMT2A
SCHEMBL27403391 0.76 KMT2A (0.64) MAPTTP53MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5010077-A Tranquilizers A/S FERROSAN (DK) 1991-04-23 US disclosed
EP-0030254-B1 BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR THERAPEUTICAL USE SCHERING AKTIENGESELLSCHAFT (DE) 1984-10-31 EP disclosed
US-4371536-A TRANQUILIZERS A/S FERROSAN (DK) 1983-02-01 US disclosed
EP-0030254-A1 Beta-carbolin-3-carboxylic acid derivatives, pharmaceutical compositions containing them and their therapeutical use SCHERING AKTIENGESELLSCHAFT (DE) 1981-06-17 EP disclosed