SCHEMBL7385263

SCHEMBL7385263

Fc1ccc(CCN2C[C@H]3CC=CC[C@H]3C2)cc1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.53
HTR2A P28223 4/20 0.46
HTR2C P28335 3/20 0.46
HTR7 P34969 3/20 0.46
HTR6 P50406 2/20 0.46
KCNJ1 P48048 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7385271 1.00 MAOA (0.53) MAOAHTR2AHTR2CHTR7HTR6
SCHEMBL7383115 0.83 HTR2A (0.49) MAOAHTR2AHTR2CHTR7HTR6
SCHEMBL7377224 0.83 SIGMAR1 (0.39) HTR2A
SCHEMBL7383109 0.83 HTR2A (0.49) MAOAHTR2AHTR2CHTR7HTR6
SCHEMBL7377219 0.83 SIGMAR1 (0.39) HTR2A
SCHEMBL7383126 0.82 SLC6A3 (0.53) MAOAHTR2AHTR2CKCNH2
SCHEMBL7383124 0.82 SLC6A3 (0.53) MAOAHTR2AHTR2CKCNH2
SCHEMBL23381594 0.80 MAOA (0.53) MAOAHTR2AHTR2CHTR7HTR6
SCHEMBL7378674 0.79 HRH3 (0.56)
SCHEMBL7378669 0.79 HRH3 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409929-A Treating psychosis, dyskinesia THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-25 US disclosed
EP-0626947-A1 HYDROISOINDOLINES AND HYDROISOQUINOLINES AS PSYCHOTROPIC DRUGS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-12-07 EP disclosed
WO-1993016047-A1 HYDROISOINDOLINES AND HYDROISOQUINOLINES AS PSYCHOTROPIC DRUGS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-08-19 WO disclosed
US-5216018-A Antidyskinetic agents DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-06-01 US disclosed