SCHEMBL7385356

SCHEMBL7385356

CC1=C(C(=O)OC(C)C)C(c2ccccc2Cl)C(S(=O)(=O)c2ccc(O)cc2)=C(C)N1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.52
ACHE P22303 1/20 0.45
NR3C2 P08235 1/20 0.44
PYGL P06737 9/20 0.43
PYGM P11217 9/20 0.43
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
MEN1 O00255 1/20 0.41
MLNR O43193 1/20 0.41
NR1I2 O75469 1/20 0.41
ABCB11 O95342 1/20 0.41
NR3C1 P04150 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7383535 0.93 CYP2C9 (0.48) ALOX15ACHENR3C2PYGLPYGM
SCHEMBL7384908 0.90 CYP2C9 (0.43) ALOX15ACHENR3C2PYGLPYGM
SCHEMBL7382716 0.90 ALOX15 (0.50) ALOX15ACHENR3C2PYGLPYGM
SCHEMBL7377019 0.89 KDM4E (0.50) MAPTKDM4ETDP1CYP1A2CYP3A4
SCHEMBL7385349 0.87 KDM4E (0.54) MAPTKDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL7382382 0.86 NR3C2 (0.45) ALOX15NR3C2MAPTKDM4ECYP1A2
SCHEMBL7376680 0.84 TBXA2R (0.48) MAPTKDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL7385182 0.84 CYP2C9 (0.49) ALOX15NR3C2MAPTKDM4ECYP1A2
SCHEMBL7376670 0.82 ALDH1A1 (0.51) MAPTKDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL7384438 0.82 CYP2C9 (0.46) ALOX15MAPTKDM4ETDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4889866-A CARDIOVASCULAR DISEASES, HYPOTENSIVE AGENTS, CONGESTIVE HEART FAILURE SYNTEX (U.S.A.) INC. (US) 1989-12-26 US disclosed