SCHEMBL7387145

SCHEMBL7387145

CCOC(=O)C1CCCCCCC(=O)C(=O)N1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.42
TSHR P16473 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
CYP2D6 P10635 1/20 0.38
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.36
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7386526 0.86 ALDH1A1 (0.37) ALDH1A1TSHRKMT2AMEN1CYP2D6
SCHEMBL7381519 0.85 LMNA (0.47) ALDH1A1TSHRKMT2AMEN1CYP2D6
SCHEMBL3066907 0.83 LMNA (0.48) ALDH1A1TSHRKMT2AMEN1CYP2D6
SCHEMBL22800174 0.79 KDM4E (0.44) ALDH1A1KMT2AMEN1KDM4ESMN1; SMN2
SCHEMBL22800767 0.79 KDM4E (0.44) ALDH1A1KMT2AMEN1KDM4ESMN1; SMN2
SCHEMBL13106060 0.78 LMNA (0.49) ALDH1A1TSHRKMT2AMEN1LMNA
SCHEMBL5992612 0.78 LMNA (0.49) ALDH1A1TSHRKMT2AMEN1LMNA
SCHEMBL15265428 0.78 LMNA (0.49) ALDH1A1TSHRKMT2AMEN1LMNA
SCHEMBL7386753 0.78 ALDH1A1 (0.40) ALDH1A1TSHRKMT2AMEN1CYP2D6
SCHEMBL7390342 0.78 TLR4 (0.43) ALDH1A1TSHRKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5426103-A Endopeptidase inhibitors; condensing macrocylic compound with a thioic acid or salt therof; possible esterification, salt formation, deslating, deprotecting, deesterifying of function-al groups CIBA-GEIGY CORPORATION (US) 1995-06-20 US disclosed
US-5244889-A Treatment of cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1993-09-14 US disclosed
EP-0544620-A1 Macrocyclic lactams as inhibitors of atrial natriuretic factors (ANF)-degrading neutral endopeptidase (NEP) CIBA-GEIGY AG (CH) 1993-06-02 EP disclosed