SCHEMBL738976

SCHEMBL738976

CCCN1CCCC(c2nc3ccccc3[nH]2)C1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.63
DRD2 P14416 1/20 0.56
DRD1 P21728 1/20 0.56
DRD4 P21917 1/20 0.56
DRD5 P21918 1/20 0.56
DRD3 P35462 1/20 0.56
KDM4E B2RXH2 3/20 0.53
PARP1 P09874 2/20 0.53
HTR2B P41595 1/20 0.50
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL666433 0.92 PARP1 (0.60) POLBDRD2PARP1HTR2BPKM
SCHEMBL14218701 0.90 POLB (0.62) POLBKDM4EHTR2BPKM
SCHEMBL9870915 0.85 HTR2B (0.56) POLBDRD2DRD1DRD4DRD5
SCHEMBL16349536 0.84 PARP1 (0.59) POLBDRD2KDM4EPARP1HTR2B
SCHEMBL17533943 0.84 PARP1 (0.59) POLBDRD2KDM4EPARP1HTR2B
SCHEMBL9869376 0.82 HTR2B (0.60) POLBKDM4EHTR2BPKM
SCHEMBL20001659 0.80 POLB (0.54) POLBKDM4EPARP1HTR2B
SCHEMBL4148001 0.79 POLB (0.56) POLBKDM4EHTR2BPKM
SCHEMBL9869744 0.79 PKM (0.56) POLBKDM4EPARP1HTR2BPKM
SCHEMBL30365989 0.79 PKM (0.56) POLBKDM4EPARP1HTR2BPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed