SCHEMBL7390477

SCHEMBL7390477

CN(C)C(=O)CNCCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.67
KCNH2 Q12809 7/20 0.56
DRD2 P14416 1/20 0.55
DRD4 P21917 1/20 0.55
OPRM1 P35372 1/20 0.55
DRD3 P35462 1/20 0.55
CA12 O43570 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
KMT2A Q03164 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
MEN1 O00255 1/20 0.47
ATM Q13315 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1867796 0.82 CYP2D6 (0.51) CYP2D6OPRM1KMT2ANPC1RAB9A
SCHEMBL68577 0.81 CYP2D6 (1.00) CYP2D6KCNH2
SCHEMBL8294306 0.81 DPP7 (0.52) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL8360505 0.80 ALDH1A1 (0.57) CA12CA2CA9KMT2ANPC1
Hydrochloric Acid SCHEMBL4228542 0.80 ALDH1A1 (0.51) CYP2D6KCNH2DRD2DRD4OPRM1
SCHEMBL157742 0.80 KEAP1 (0.59) CA12CA2CA9SIGMAR1GAA
SCHEMBL28813550 0.79 CYP2D6 (0.59) CYP2D6KCNH2
Hydrochloric Acid SCHEMBL27975380 0.78 KCNH2 (0.59) CYP2D6KCNH2
SCHEMBL27759805 0.78 KEAP1 (0.57) CA12CA2CA9SIGMAR1GAA
Hydrochloric Acid SCHEMBL10493762 0.78 MAPT (0.59) CA12CA2CA9SIGMAR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0589445-B1 Renin Inhibiting N-(2-Amino-2-oxoethyl)Butanediamide Derivatives BIO MEGA BOEHRINGER INGELHEIM (CA) 1997-01-15 EP disclosed
US-5541163-A HYPOTENSIVE AGENTS BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1996-07-30 US disclosed
WO-1994007846-A1 RENIN INHIBITING N-(2-AMINO-2-OXOETHYL)BUTANEDIAMIDE DERIVATIVES BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1994-04-14 WO disclosed
EP-0589445-A1 Renin Inhibiting N-(2-Amino-2-oxoethyl)Butanediamide Derivatives BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1994-03-30 EP disclosed