SCHEMBL7393752

SCHEMBL7393752

CCOc1cc2c(cc1OC)/C(=C(/C#N)CCCN1CCCC1)NC1CCCCC21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EHMT2 Q96KQ7 8/20 0.35
NSD2 O96028 7/20 0.34
LMNA P02545 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
CYP2D6 P10635 1/20 0.34
ADRA2C P18825 1/20 0.34
OPRK1 P41145 1/20 0.34
KCNH2 Q12809 1/20 0.34
EBP Q15125 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
KMT5A Q9NQR1 2/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444417 1.00 EHMT2 (0.35) EHMT2NSD2LMNAHTR1AADRA2A
SCHEMBL7393757 1.00 EHMT2 (0.35) EHMT2NSD2LMNAHTR1AADRA2A
SCHEMBL7403389 0.99 EHMT2 (0.36) EHMT2NSD2LMNAHTR1AADRA2A
SCHEMBL7403386 0.99 EHMT2 (0.36) EHMT2NSD2LMNAHTR1AADRA2A
SCHEMBL7445293 0.99 EHMT2 (0.36) EHMT2NSD2LMNAHTR1AADRA2A
SCHEMBL7447087 0.95 CHEK1 (0.34) EHMT2NSD2HTR1APDE4APDE4B
SCHEMBL7447103 0.95 CHEK1 (0.34) EHMT2NSD2HTR1APDE4APDE4B
SCHEMBL7447093 0.95 CHEK1 (0.34) EHMT2NSD2HTR1APDE4APDE4B
SCHEMBL7400407 0.94 CHEK1 (0.37) NSD2LMNABCHEACHECHEK1
SCHEMBL7400404 0.94 CHEK1 (0.37) NSD2LMNABCHEACHECHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001064648-A1 ISOQUINOLINE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-07 WO claimed
WO-2001064648-A1 ISOQUINOLINE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-07 WO disclosed