SCHEMBL7447103

SCHEMBL7447103

CCOc1cc2c(cc1OC)C(=C(C#N)CCCN1CCN(C)CC1)NC1CCCCC21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
EHMT2 Q96KQ7 5/20 0.33
NSD2 O96028 4/20 0.33
HTR1A P08908 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
HTR2B P41595 1/20 0.33
WEE2 P0C1S8 1/20 0.32
WEE1 P30291 1/20 0.32
PKMYT1 Q99640 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447093 1.00 CHEK1 (0.34) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL7447087 1.00 CHEK1 (0.34) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL7393752 0.95 EHMT2 (0.35) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL7393757 0.95 EHMT2 (0.35) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL7444417 0.95 EHMT2 (0.35) CHEK1PDE4APDE4BPDE4CPDE4D
SCHEMBL7403386 0.94 EHMT2 (0.36) CHEK1EHMT2NSD2HTR1A
SCHEMBL7403389 0.94 EHMT2 (0.36) CHEK1EHMT2NSD2HTR1A
SCHEMBL7445293 0.94 EHMT2 (0.36) CHEK1EHMT2NSD2HTR1A
SCHEMBL7400404 0.92 CHEK1 (0.37) CHEK1NSD2
SCHEMBL7400407 0.92 CHEK1 (0.37) CHEK1NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001064648-A1 ISOQUINOLINE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-07 WO disclosed