SCHEMBL7445293

SCHEMBL7445293

CCOc1cc2c(cc1OC)C(=C(C#N)CCCN1CCCCC1)NC1CCCCC21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EHMT2 Q96KQ7 7/20 0.36
NSD2 O96028 6/20 0.34
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
CHEK1 O14757 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
LMNA P02545 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
CYP2D6 P10635 1/20 0.33
ADRA2C P18825 1/20 0.33
OPRK1 P41145 1/20 0.33
KCNH2 Q12809 1/20 0.33
EBP Q15125 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
CACNA1C Q13936 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7403386 1.00 EHMT2 (0.36) EHMT2NSD2BCHEACHECHEK1
SCHEMBL7403389 1.00 EHMT2 (0.36) EHMT2NSD2BCHEACHECHEK1
SCHEMBL7444417 0.99 EHMT2 (0.35) EHMT2NSD2BCHEACHECHEK1
SCHEMBL7393752 0.99 EHMT2 (0.35) EHMT2NSD2BCHEACHECHEK1
SCHEMBL7393757 0.99 EHMT2 (0.35) EHMT2NSD2BCHEACHECHEK1
SCHEMBL7447087 0.94 CHEK1 (0.34) EHMT2NSD2CHEK1HTR1A
SCHEMBL7447103 0.94 CHEK1 (0.34) EHMT2NSD2CHEK1HTR1A
SCHEMBL7447093 0.94 CHEK1 (0.34) EHMT2NSD2CHEK1HTR1A
SCHEMBL7400404 0.93 CHEK1 (0.37) NSD2BCHEACHECHEK1LMNA
SCHEMBL7400407 0.93 CHEK1 (0.37) NSD2BCHEACHECHEK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001064648-A1 ISOQUINOLINE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-07 WO claimed
WO-2001064648-A1 ISOQUINOLINE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-07 WO disclosed