SCHEMBL7394236

SCHEMBL7394236

COc1ccc(C2CCNCCS2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.74
MAP2K1 Q02750 1/20 0.58
MAOB P27338 5/20 0.52
KDM1A O60341 1/20 0.48
TDP1 Q9NUW8 1/20 0.46
HTR2C P28335 2/20 0.43
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
HRH1 P35367 2/20 0.41
KCNH2 Q12809 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ADRB1 P08588 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1636984 0.85 MAOA (1.00) MAOAMAP2K1MAOBKDM1AHTR2C
SCHEMBL6331656 0.81 MAOB (0.52) MAOAMAP2K1MAOBKDM1AHRH1
SCHEMBL9359327 0.80 MAOA (0.58) MAOAMAP2K1MAOBKDM1AKMT2A
SCHEMBL6610340 0.78 MAOA (0.57) MAOAMAP2K1MAOBKDM1AKMT2A
SCHEMBL31322216 0.78 SLC18A3 (0.53) MAOAMAOBKDM1AHTR2CHRH1
SCHEMBL239790 0.75 HTR2C (0.64) MAOAMAOBKDM1ATDP1HTR2C
Hydrochloric Acid SCHEMBL2800981 0.74 HTR2C (0.65) MAOAMAOBKDM1ATDP1HTR2C
SCHEMBL6331476 0.74 MAP2K1 (1.00) MAOAMAP2K1MAOBKMT2A
SCHEMBL7399263 0.73 MAOA (0.51) MAOAMAP2K1HTR2CKMT2AALDH1A1
SCHEMBL2084131 0.71 MAPT (0.66) MAOAMAP2K1MAOBKDM1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5206233-A Antidepressants, antiischemic agents WARNER-LAMBERT COMPANY (US) 1993-04-27 US claimed
WO-1993004053-A1 SUBSTITUTED THIAZEPINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
US-5206233-A Antidepressants, antiischemic agents WARNER-LAMBERT COMPANY (US) 1993-04-27 US disclosed
WO-1993004053-A1 SUBSTITUTED THIAZEPINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed