SCHEMBL7399263

SCHEMBL7399263

COc1ccc(C2CCN(C)CCS2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.51
MAP2K1 Q02750 1/20 0.47
DRD2 P14416 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RYR2 Q92736 1/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
RAB9A P51151 1/20 0.41
USP2 O75604 1/20 0.40
BRD4 O60885 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KDM4E B2RXH2 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401016 0.81 DRD2 (0.66) MAOAMAP2K1DRD2BRD4
SCHEMBL7403885 0.81 LSS (0.47) DRD2HTR2AHTR2CL3MBTL1
SCHEMBL7402278 0.81 DRD2 (0.50) MAOAMAP2K1DRD2KMT2AALDH1A1
SCHEMBL7398714 0.81 MAOA (0.48) MAOAMAP2K1DRD2KMT2AALDH1A1
SCHEMBL7402707 0.80 BRD4 (0.54) BRD4
SCHEMBL7398210 0.80 KDM4E (0.47) MAOAMAP2K1KMT2AALDH1A1GAA
Hydrochloric Acid SCHEMBL7398529 0.79 LSS (0.46) DRD2HTR2AHTR2CL3MBTL1
SCHEMBL9359327 0.78 MAOA (0.58) MAOAMAP2K1DRD2KMT2AALDH1A1
SCHEMBL6610340 0.77 MAOA (0.57) MAOAMAP2K1KMT2AALDH1A1PTGS1
SCHEMBL4403006 0.76 DRD2 (0.68) DRD2ALDH1A1GAAHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5206233-A Antidepressants, antiischemic agents WARNER-LAMBERT COMPANY (US) 1993-04-27 US claimed
WO-1993004053-A1 SUBSTITUTED THIAZEPINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
US-5206233-A Antidepressants, antiischemic agents WARNER-LAMBERT COMPANY (US) 1993-04-27 US disclosed
WO-1993004053-A1 SUBSTITUTED THIAZEPINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed