SCHEMBL7397116

SCHEMBL7397116

N#Cc1cccc(O)c1.[NaH]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.52
CA12 O43570 3/20 0.50
CA2 P00918 3/20 0.50
CA9 Q16790 3/20 0.50
ALDH1A1 P00352 3/20 0.50
CA14 Q9ULX7 2/20 0.50
P4HB P07237 2/20 0.50
LMNA P02545 1/20 0.50
CYP3A4 P08684 1/20 0.50
CA5A P35218 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
CA3 P07451 1/20 0.48
CA6 P23280 1/20 0.48
TSHR P16473 1/20 0.46
GSK3B P49841 2/20 0.44
CLK4 Q9HAZ1 1/20 0.44
XDH P47989 1/20 0.43
SLC22A12 Q96S37 1/20 0.43
MAPT P10636 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1330201 0.98
SCHEMBL29566889 0.98
SCHEMBL51546 0.98
Hydrochloric Acid SCHEMBL28758837 0.95 ENPP2 (0.52) ENPP2CA12CA2CA9ALDH1A1
SCHEMBL27941360 0.89 CA12 (0.50) ENPP2CA12CA2CA9P4HB
Butane SCHEMBL27795956 0.87 ENPP2 (0.46) ENPP2CA12CA2CA9ALDH1A1
SCHEMBL28140796 0.86 ENPP2 (0.48) ENPP2CA12CA2CA9ALDH1A1
SCHEMBL1029016 0.85 HSD17B1 (0.58) ENPP2P4HBCYP3A4CLK4XDH
SCHEMBL30165928 0.85 HSD17B1 (0.58) ENPP2P4HBCYP3A4CLK4XDH
Benzonitrile SCHEMBL28338020 0.84 TSHR (0.64) ENPP2CA12CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123933-A1 2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]chromane as CNS active agent MERCK PATENT GmbH (DE) 2001-08-16 EP disclosed
US-5767132-A CENTRAL NERVOUS SYSTEM MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-06-16 US disclosed
EP-0707007-A1 Amino(thio)ether derivatives as CNS active agents MERCK PATENT GmbH (DE) 1996-04-17 EP disclosed
US-4031232-A 1-Alkyl-2-(phenoxymethyl)-5-nitro-imidazoles and process for their manufacture HOECHST AKTIENGESELLSCHAFT (DT) 1977-06-21 US disclosed