SCHEMBL7397389

SCHEMBL7397389

COc1ccc(N2CCN(CCC3CCCc4ccccc43)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 5/20 0.66
DRD2 P14416 3/20 0.66
HTR1A P08908 2/20 0.66
HTR1D P28221 1/20 0.66
HTR2A P28223 1/20 0.66
SIGMAR1 Q99720 5/20 0.56
ADRA1A P35348 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7399648 0.99 DRD4 (0.64) DRD4DRD2HTR1AHTR1DHTR2A
SCHEMBL7397854 0.93 DRD4 (0.68) DRD4DRD2HTR1AHTR1DHTR2A
Hydrochloric Acid SCHEMBL8185604 0.92 DRD4 (0.67) DRD4DRD2HTR1AHTR1DHTR2A
SCHEMBL7403278 0.85 ALDH1A1 (0.59) DRD4DRD2HTR1AHTR2ASIGMAR1
Hydrochloric Acid SCHEMBL7401194 0.84 ALDH1A1 (0.58) DRD4DRD2HTR1AHTR2ASIGMAR1
SCHEMBL7406795 0.83 SIGMAR1 (0.47) DRD4DRD2HTR1AHTR1DHTR2A
Hydrochloric Acid SCHEMBL7401132 0.82 SIGMAR1 (0.47) DRD4DRD2HTR1AHTR1DHTR2A
SCHEMBL7407464 0.82 DRD2 (0.88) DRD4DRD2HTR1AHTR1DHTR2A
SCHEMBL7402337 0.81 DRD2 (0.48) DRD4DRD2HTR1AHTR1DHTR2A
Hydrochloric Acid SCHEMBL7398494 0.81 DRD4 (0.56) DRD4DRD2HTR1AHTR1DHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737189-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1996-10-16 EP claimed
WO-1995018118-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS THE UPJOHN COMPANY (US) 1995-07-06 WO claimed
US-6133446-A Heterocyclic compounds for the treatment of CNS and cardiovascular disorders PHARMACIA & UPJOHN COMPANY (US) 2000-10-17 US disclosed
EP-0737189-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1996-10-16 EP disclosed
WO-1995018118-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS THE UPJOHN COMPANY (US) 1995-07-06 WO disclosed