SCHEMBL7397491

SCHEMBL7397491

N[C@H](CC(=O)OC(=O)c1ccc(OCCN2CCCC2)cc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 10/20 0.52
LTA4H P09960 2/20 0.52
KCNH2 Q12809 2/20 0.52
KDM4E B2RXH2 1/20 0.51
PSMB1 P20618 5/20 0.47
PSMB5 P28074 4/20 0.47
PSMB2 P49721 2/20 0.47
HTR1A P08908 1/20 0.45
HTR7 P34969 1/20 0.45
ESR1 P03372 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402237 0.88 ESR1 (0.48) HRH3LTA4HKCNH2HTR1AHTR7
SCHEMBL7397850 0.87 EPHX2 (0.47) HRH3KDM4E
Hydrochloric Acid SCHEMBL7488066 0.84 ITGB3 (0.59) ESR1
SCHEMBL7399207 0.81 ITGB3 (0.55)
SCHEMBL8458587 0.81 SLC1A3 (0.47) KDM4E
SCHEMBL7487574 0.80 ITGB3 (0.48)
SCHEMBL7398725 0.80 ITGB3 (0.46) HRH3LTA4HKCNH2KDM4EHTR1A
SCHEMBL7399762 0.80 ITGB3 (0.50)
SCHEMBL7397774 0.80 ITGB3 (0.44)
SCHEMBL7398498 0.80 TBXAS1 (0.53) KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648368-A ANTICOAGULANTS MERCK & CO., INC. (US) 1997-07-15 US disclosed
EP-0673247-A4 FIBRINOGEN RECEPTOR ANTAGONISTS. MERCK & CO INC (US) 1996-05-01 EP disclosed
EP-0673247-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1995-09-27 EP disclosed
WO-1994012181-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-06-09 WO disclosed