SCHEMBL7398207

SCHEMBL7398207

O=C=CN(CC(=O)O)OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
MAPK1 P28482 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PAM P19021 1/20 0.40
HCAR2 Q8TDS4 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAOB P27338 3/20 0.37
LMNA P02545 2/20 0.36
AKR1B1 P15121 1/20 0.36
KEAP1 Q14145 1/20 0.36
CASP1 P29466 1/20 0.36
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6566174 0.82 ALDH1A1 (0.44) ALDH1A1MAPK1L3MBTL1PAMHCAR2
SCHEMBL7587208 0.74 ALDH1A1 (0.47) ALDH1A1MAPK1L3MBTL1HCAR2SLC6A2
SCHEMBL6271777 0.73 ALDH1A1 (0.46) ALDH1A1MAPK1L3MBTL1HCAR2SLC6A2
SCHEMBL27739393 0.73 ALDH1A1 (0.46) ALDH1A1MAPK1L3MBTL1HCAR2SLC6A2
SCHEMBL11330873 0.71 ALDH1A1 (0.48) ALDH1A1MAPK1L3MBTL1SLC6A2SLC6A3
SCHEMBL30803699 0.71 ALDH1A1 (0.44) ALDH1A1MAPK1L3MBTL1HCAR2SLC6A2
SCHEMBL8592588 0.71 ALDH1A1 (0.40) ALDH1A1MAPK1L3MBTL1HCAR2SLC6A2
SCHEMBL5370663 0.70 ALDH1A1 (0.43) ALDH1A1MAPK1L3MBTL1SLC6A2SLC6A3
SCHEMBL8740511 0.70 SLC1A3 (0.41) ALDH1A1MAPK1L3MBTL1HCAR2SLC6A2
SCHEMBL6951407 0.70 HTT (0.44) ALDH1A1MAPK1HCAR2SLC6A3KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994013636-A1 NEW SUBSTITUTED AZETIDINONES AS ANTI-INFLAMMATORY AND ANTIDEGENERATIVE AGENTS MERCK & CO., INC. (US) 1994-06-23 WO disclosed
EP-0144103-B1 Methods and compositions for preparation of H-ARG-X-Z-Y-TYR-R ORTHO PHARMA CORP (US) 1993-12-29 EP disclosed
EP-0144103-A2 Methods and compositions for preparation of H-ARG-X-Z-Y-TYR-R ORTHO PHARMACEUTICAL CORPORATION (US) 1985-06-12 EP disclosed