SCHEMBL7399324

SCHEMBL7399324

CC(C)C[C@@H](C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCN1CCCCC1)N(C)CC1CCCCC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.48
CTSK P43235 4/20 0.47
TACR2 P21452 5/20 0.46
PLG P00747 1/20 0.45
PRSS1 P07477 1/20 0.45
PRSS2 P07478 1/20 0.45
PRSS3 P35030 1/20 0.45
CACNA1B Q00975 4/20 0.45
PSMB1 P20618 1/20 0.45
PSMB8 P28062 1/20 0.45
PSMB9 P28065 1/20 0.45
PSMB5 P28074 1/20 0.45
YAP1 P46937 2/20 0.44
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
CTSL P07711 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7398380 0.89 CTSS (0.53) CTSSCTSKTACR2CACNA1BPSMB8
SCHEMBL7401303 0.89 CTSS (0.50) CTSSCTSKTACR2CACNA1BPSMB8
SCHEMBL7408154 0.89 CTSS (0.54) CTSSCTSKTACR2PSMB8PSMB9
SCHEMBL7446475 0.88 CTSS (0.51) CTSSCTSKTACR2CACNA1BPSMB8
SCHEMBL7402336 0.87 CACNA1B (0.55) CACNA1BYAP1
SCHEMBL8193256 0.87 CTSS (0.48) CTSSCTSKTACR2CACNA1BPSMB8
SCHEMBL7504668 0.87 CTSS (0.51) CTSSCTSKTACR2PLGPRSS1
SCHEMBL8193049 0.86 CTSS (0.48) CTSSCTSKTACR2CACNA1BYAP1
SCHEMBL7406386 0.85 CACNA1B (0.51) CACNA1BYAP1
SCHEMBL7405818 0.85 CACNA1B (0.49) CACNA1BPSMB1PSMB8PSMB9PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed