SCHEMBL7401303

SCHEMBL7401303

CC(C)CCN(C)[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCN1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.50
CACNA1B Q00975 4/20 0.48
TACR2 P21452 6/20 0.48
CTSK P43235 1/20 0.45
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
PSMB8 P28062 1/20 0.44
PSMB9 P28065 1/20 0.44
PSMB5 P28074 1/20 0.44
PSMB10 P40306 1/20 0.44
PSMB2 P49721 1/20 0.44
CTSL P07711 1/20 0.44
IL1RN P18510 1/20 0.43
ERAP2 Q6P179 1/20 0.43
ERAP1 Q9NZ08 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446475 0.99 CTSS (0.51) CTSSCACNA1BTACR2CTSKITGB3
SCHEMBL7405180 0.93 TACR2 (0.57) TACR2PSMB8PSMB9PSMB5PSMB10
SCHEMBL7398380 0.91 CTSS (0.53) CTSSCACNA1BTACR2CTSKITGB3
SCHEMBL5833220 0.91 CTSS (0.47) CTSSCACNA1BTACR2CTSKITGB3
SCHEMBL7408154 0.91 CTSS (0.54) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL5833014 0.89 PLG (0.46) CTSSCACNA1BTACR2CTSKITGB3
SCHEMBL7399324 0.89 CTSS (0.48) CTSSCACNA1BTACR2CTSKITGB3
SCHEMBL8193256 0.89 CTSS (0.48) CTSSCACNA1BTACR2CTSKITGB3
SCHEMBL5833276 0.89 TACR2 (0.44) CTSSCACNA1BTACR2ITGB3ITGA2B
SCHEMBL8193049 0.88 CTSS (0.48) CTSSCACNA1BTACR2CTSKITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863919-B1 SUPPORTED CATALYST CONTAINING TETHERED CATION FORMING ACTIVATOR DOW CHEMICAL CO (US) 2000-11-15 EP disclosed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed