SCHEMBL7399556

SCHEMBL7399556

COC(=O)c1cc(Cl)cc(C2CC=CCC2)c1O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
TP53 P04637 2/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SLC6A3 Q01959 5/20 0.36
SERPINH1 P50454 1/20 0.35
ABL1 P00519 1/20 0.35
ALDH1A1 P00352 2/20 0.34
PTGDR Q13258 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
GAA P10253 2/20 0.34
HTT P42858 1/20 0.34
NR4A2 P43354 1/20 0.34
OPRK1 P41145 1/20 0.34
ACLY P53396 1/20 0.33
SLC6A4 P31645 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416449 0.84 AKR1C2 (0.46) LMNATP53TSHRSMN1; SMN2ALDH1A1
SCHEMBL7413453 0.79 LMNA (0.41) LMNATP53TSHRSMN1; SMN2ALDH1A1
SCHEMBL7396665 0.74 SMN1; SMN2 (0.34) LMNATP53TSHRSMN1; SMN2ALDH1A1
SCHEMBL10546858 0.73 SERPINH1 (0.38) LMNATSHRSMN1; SMN2SLC6A3SERPINH1
SCHEMBL27201936 0.71 GAA (0.45) LMNATSHRSLC6A3ABL1ALDH1A1
SCHEMBL30689803 0.71 GAA (0.45) LMNATSHRSLC6A3ABL1ALDH1A1
SCHEMBL19612159 0.70 KDM4E (0.43) TSHRSMN1; SMN2SLC6A3SERPINH1ABL1
SCHEMBL3224195 0.70 ABL1 (0.45) LMNATSHRSLC6A3SERPINH1ABL1
SCHEMBL855750 0.69 LMNA (0.52) LMNATSHRSMN1; SMN2SLC6A3SERPINH1
SCHEMBL423691 0.69 AKR1C4 (0.60) TSHRSLC6A3SERPINH1ABL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-H1406-H Process for preparing dibenzofurans via catalytic heteroannulation RHONE POULENC RORER PHARMACEUTICALS INC. (US) 1995-01-03 US disclosed
US-5288731-A Antiemetics, antiserotonine agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-02-22 US disclosed
US-5246942-A Central nervous system, anti-emetic and gastric prokinetic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1993-09-21 US disclosed
EP-0559656-A1 PROCESS FOR PREPARING MULTICYCLIC OXY-CONTAINING RING COMPONENTS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1993-09-15 EP disclosed
EP-0494140-A4 DIBENZOFURANCARBOXAMIDES 1992-09-02 EP disclosed
EP-0494140-A1 DIBENZOFURANCARBOXAMIDES RORER INTERNATIONAL (HOLDINGS), INC. (US) 1992-07-15 EP disclosed
WO-1992009592-A1 PROCESS FOR PREPARING MULTICYCLIC OXY-CONTAINING RING COMPONENTS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1992-06-11 WO disclosed
WO-1992009284-A1 2,6-METHANO-2H-1-BENZOXOCINCARBOXAMIDES AS 5-HT3-ANTAGONISTS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS), INC. (US) 1992-06-11 WO disclosed
WO-1991004738-A1 DIBENZOFURANCARBOXAMIDES RORER INTERNATIONAL (HOLDINGS), INC. (US) 1991-04-18 WO disclosed
WO-1989010364-A1 DIBENZOFURANCARBOXAMIDES RORER INTERNATIONAL (OVERSEAS) INC. (US) 1989-11-02 WO disclosed
EP-0339950-A2 Dibenzofurancarboxamides, their use as pharmaceutical agents, a composition containing the same, and a process for the preparation thereof RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1989-11-02 EP disclosed