SCHEMBL7416449

SCHEMBL7416449

O=C(O)c1cc(Cl)cc(C2CC=CCC2)c1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 2/20 0.46
AKR1C1 Q04828 2/20 0.46
AKR1C3 P42330 2/20 0.46
AKR1C4 P17516 1/20 0.46
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CYP3A4 P08684 1/20 0.35
TP53 P04637 2/20 0.34
HTT P42858 2/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
ACMSD Q8TDX5 2/20 0.34
SERPINE1 P05121 2/20 0.33
KDM4C Q9H3R0 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399556 0.84 LMNA (0.38) ALDH1A1TP53HTTLMNAGAA
SCHEMBL9249778 0.80 AKR1C4 (0.53) AKR1C2AKR1C1AKR1C3AKR1C4ALDH1A1
SCHEMBL9510268 0.77 ALDH1A1 (0.41) AKR1C3ALDH1A1HPGDHSD17B10CA1
SCHEMBL4357324 0.71 RAB9A (0.43) AKR1C3ALDH1A1HPGDCA1CA2
SCHEMBL8629633 0.69 MAPT (0.32) AKR1C3MAPT
SCHEMBL10369790 0.68 KDM4C (0.44) ALDH1A1KDM4CKDM4EMEN1MAPT
SCHEMBL6289089 0.66 AKR1C2 (0.64) AKR1C2AKR1C1AKR1C3AKR1C4ALDH1A1
SCHEMBL4862551 0.65 AKR1C2 (0.69) AKR1C2AKR1C1AKR1C3AKR1C4ALDH1A1
SCHEMBL29375230 0.65 AKR1C2 (1.00) AKR1C2AKR1C1AKR1C3AKR1C4ALDH1A1
SCHEMBL184603 0.65 AKR1C2 (1.00) AKR1C2AKR1C1AKR1C3AKR1C4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5288731-A Antiemetics, antiserotonine agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1994-02-22 US disclosed
WO-1992009284-A1 2,6-METHANO-2H-1-BENZOXOCINCARBOXAMIDES AS 5-HT3-ANTAGONISTS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS), INC. (US) 1992-06-11 WO disclosed