SCHEMBL7399570

SCHEMBL7399570

Cn1c(=O)c2[nH]c(/C=C/c3cccc([N+](=O)[O-])c3)nc2n(C)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MITF O75030 1/20 0.62
ADORA2B P29275 2/20 0.54
MEN1 O00255 1/20 0.54
LMNA P02545 1/20 0.54
MAPT P10636 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54
KMT2A Q03164 1/20 0.54
MCL1 Q07820 1/20 0.54
PTK2B Q14289 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399571 1.00 MITF (0.62) MITFADORA2BMEN1LMNAMAPT
SCHEMBL7731353 0.84 ADORA3 (0.55) ADORA2B
SCHEMBL7731346 0.84 ADORA3 (0.55) ADORA2B
SCHEMBL7311779 0.82 SMN1; SMN2 (0.57) MEN1LMNAMAPTHTTRAB9A
SCHEMBL7311794 0.82 SMN1; SMN2 (0.57) MEN1LMNAMAPTHTTRAB9A
SCHEMBL7399777 0.82
SCHEMBL7399778 0.82
SCHEMBL7400082 0.81
SCHEMBL7400086 0.81
SCHEMBL7395581 0.80 MAOA (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861405-A A2-SELECTIVE ADENOSINE RECEPTOR ANTAGONIST AS ANTIDEPRESSANTS AND CNS STIMULANTS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1999-01-19 US disclosed
WO-1994025462-A1 8-SUBSTITUTED 1,3,7-TRIALKYL-XANTHINE DERIVATIVES AS A2-SELECTIVE ADENOSINE RECEPTOR ANTAGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY THE (US) 1994-11-10 WO disclosed