SCHEMBL7399760

SCHEMBL7399760

CC1(C)CCc2[nH]cc(C(=O)Nc3ccccc3F)c2C1=O

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.56
ROCK1 Q13464 1/20 0.56
LMNA P02545 2/20 0.51
NPC1 O15118 5/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 6/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
RORC P51449 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394552 0.86 ROCK2 (0.49) ROCK2ROCK1LMNANPC1HTT
SCHEMBL7397319 0.84 ROCK2 (0.68) ROCK2ROCK1LMNANPC1HTT
SCHEMBL7392152 0.83 ROCK2 (0.47) ROCK2ROCK1LMNANPC1SMN1; SMN2
SCHEMBL7395738 0.83 ROCK2 (0.47) ROCK2ROCK1NPC1SMN1; SMN2RAB9A
SCHEMBL7369380 0.82 ROCK2 (0.63) ROCK2ROCK1LMNANPC1SMN1; SMN2
SCHEMBL7400004 0.81 ROCK2 (0.45) ROCK2ROCK1LMNAHTTMEN1
SCHEMBL6778444 0.81 LMNA (0.52) LMNANPC1SMN1; SMN2HTTRAB9A
SCHEMBL7395661 0.81 ROCK2 (0.57) ROCK2ROCK1LMNANPC1HTT
SCHEMBL7359535 0.79 LMNA (0.55) LMNANPC1SMN1; SMN2HTTRAB9A
SCHEMBL4902848 0.79 LMNA (0.55) LMNANPC1SMN1; SMN2HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998002420-A9 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS 1998-04-23 WO claimed
WO-1998002420-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO claimed
US-5925770-A GAMMA-AMINOBUTYRIC ACID DERIVATIVES FOR DIAGNOSIS OR TREATMENT OF ANXIETY, SLEEP DISORDERS, SEIZURES, OVERDOSES OF BENZODIAZEPINE TYPE DRUGS, COGNITION ACTIVATORS NEUROGEN CORPORATION (US) 1999-07-20 US disclosed
US-5750702-A Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands NEUROGEN CORPORATION (US) 1998-05-12 US disclosed
WO-1998002420-A9 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS 1998-04-23 WO disclosed
WO-1998002420-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO disclosed