SCHEMBL7399776

SCHEMBL7399776

CC(=O)Nc1cc[c]cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
ALDH1A1 P00352 4/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
POLB P06746 3/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
PKM P14618 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 2/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2489381 0.85 HDAC1 (0.42) HDAC1HDAC6CA1CA2CA9
SCHEMBL27943823 0.84 POLB (0.47) HDAC1CA1CA2CA9ALDH1A1
SCHEMBL5831442 0.82 ALDH1A1 (0.44) CA1CA2CA9ALDH1A1HPGD
SCHEMBL10803626 0.81 NPC1 (0.43) HDAC1HDAC6CA1CA2CA9
SCHEMBL6205970 0.79 ALDH1A1 (0.55) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL28297471 0.79 POLB (0.52) HDAC1CA1CA2CA9ALDH1A1
SCHEMBL21357 0.78 CA1 (0.45) CA1CA2CA9ALDH1A1HPGD
SCHEMBL27193000 0.77 TGM2 (0.46) ALDH1A1LMNACYP2C19
SCHEMBL27544601 0.77 CYP17A1 (0.44) NPC1RAB9APOLBLMNA
SCHEMBL220305 0.77 ALDH1A1 (0.57) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134708-A1 THIAZOLOPYRIDYL AMIDE DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS BEIGENE , LTD. (KY) 2023-07-20 WO disclosed
US-6043263-A (2,3-dihydrobenzofuranyl)-thiazoles as phosphodiesterase inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-03-28 US disclosed
EP-0941226-A1 (2,3-DIHYDROBENZOFURANYL)-THIAZOLES AS PHOSPHODIESTERASE INHIBITORS Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-09-15 EP disclosed
EP-0510440-B1 Positive-working radiation-sensitive composition and radiation-sensitive recording material produced therewith CLARIANT GMBH (DE) 1999-01-13 EP disclosed
WO-1998021207-A1 (2,3-DIHYDROBENZOFURANYL)-THIAZOLES AS PHOSPHODIESTERASE INHIBITORS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-05-22 WO disclosed
WO-1998008844-A1 THIAZOLE DERIVATIVES USEFUL AS SELECTIVE INHIBITORS OF PDE-IV BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-03-05 WO disclosed
EP-0519298-B1 Radiation-sensitive sulfonic acid esters and their use HOECHST AG (DE) 1995-09-13 EP disclosed
US-5442061-A Recording, photoresists, printing plates HOECHST AKTIENGESELLSCHAFT (DE) 1995-08-15 US disclosed
EP-0510443-B1 Negative-working radiation-sensitive composition and radiation-sensitive recording material produced therewith HOECHST AG (DE) 1995-03-22 EP disclosed
US-5364734-A Sulfonated triazines HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-15 US disclosed
US-5298364-A Negative photoresists, acid crosslinking HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-29 US disclosed
US-5286867-A Substituted 1-sulfonyloxy-2-pyridones and process for preparing them HOECHST AKTIENGESELLSCHAFT (DE) 1994-02-15 US disclosed
US-5230985-A NEGATIVE-WORKING RADIATION-SENSITIVE MIXTURES, AND RADIATION-SENSITIVE RECORDING MATERIAL PRODUCED WITH THESE MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1993-07-27 US disclosed
US-5229254-A Photoresists, printing plates, sulfonic acid generators HOECHST AKTIENGESELLSCHAFT (DE) 1993-07-20 US disclosed
EP-0519298-A1 Radiation-sensitive sulfonic acid esters and their use HOECHST AKTIENGESELLSCHAFT (DE) 1992-12-23 EP disclosed
EP-0519299-A1 Positive-working radiation-sensitive composition and radiation-sensitive recording material produced therewith HOECHST AKTIENGESELLSCHAFT (DE) 1992-12-23 EP disclosed
EP-0510442-A1 Substituted 1-sulfonyloxy-2-pyridones, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1992-10-28 EP disclosed
EP-0510443-A1 Negative-working radiation-sensitive composition and radiation-sensitive recording material produced therewith HOECHST AKTIENGESELLSCHAFT (DE) 1992-10-28 EP disclosed
EP-0510440-A1 Positive-working radiation-sensitive composition and radiation-sensitive recording material produced therewith HOECHST AKTIENGESELLSCHAFT (DE) 1992-10-28 EP disclosed