Phosphine

Phosphine

SCHEMBL7400153

CC(C)C(c1ccccc1)C(Br)(c1ccccc1)c1ccccc1.P

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.39
TAAR1 Q96RJ0 3/20 0.38
AOC3 Q16853 1/20 0.35
RIPK1 Q13546 1/20 0.35
ADRA2A P08913 1/20 0.34
ADRA2C P18825 1/20 0.34
LMNA P02545 1/20 0.34
HIF1A Q16665 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MC4R P32245 1/20 0.34
CYP1A2 P05177 1/20 0.34
KCNN4 O15554 2/20 0.33
KIF11 P52732 1/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosphine SCHEMBL9506700 0.77 CYP2D6 (0.41) CYP2D6TAAR1AOC3RIPK1ADRA2A
SCHEMBL10360017 0.77 RIPK1 (0.45) CYP2D6TAAR1AOC3RIPK1ADRA2A
Bromide SCHEMBL7400155 0.75 CYP2D6 (0.36) CYP2D6TAAR1AOC3RIPK1ADRA2A
SCHEMBL8097006 0.73 TAAR1 (0.40) CYP2D6TAAR1AOC3RIPK1ADRA2A
SCHEMBL14367700 0.73 TAAR1 (0.40) CYP2D6TAAR1AOC3RIPK1ADRA2A
SCHEMBL8097109 0.73 TAAR1 (0.40) CYP2D6TAAR1AOC3RIPK1ADRA2A
SCHEMBL17084089 0.71 SLC6A4 (0.42) TAAR1AOC3RIPK1ADRA2AADRA2C
SCHEMBL17084162 0.71 SLC6A4 (0.42) TAAR1AOC3RIPK1ADRA2AADRA2C
SCHEMBL16133820 0.71 RIPK1 (0.41) CYP2D6TAAR1AOC3RIPK1ADRA2A
SCHEMBL16133821 0.71 RIPK1 (0.41) CYP2D6TAAR1AOC3RIPK1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0587767-A1 HYDROXYAZIDO DERIVATIVES AND RELATED COMPOUNDS AS RENIN INHIBITORS SRI INTERNATIONAL (US) 1994-03-23 EP disclosed
US-5268361-A Containing amide groups SRI INTERNATIONAL (US) 1993-12-07 US disclosed
WO-1992021696-A1 HYDROXYAZIDO DERIVATIVES AND RELATED COMPOUNDS AS RENIN INHIBITORS SRI INTERNATIONAL (US) 1992-12-10 WO disclosed