SCHEMBL7400381

SCHEMBL7400381

N[C@@H](Cc1ccc(C(=O)N2CCOCC2)cc1)C(=O)NC(C=Cc1ccc(Cl)s1)CCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 9/20 0.50
CTSB P07858 7/20 0.48
CTSS P25774 4/20 0.43
CTSK P43235 3/20 0.43
CTSH P09668 2/20 0.43
CTSC P53634 2/20 0.43
MASP2 O00187 1/20 0.41
F2 P00734 1/20 0.41
GAA P10253 1/20 0.41
ACACB O00763 1/20 0.40
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354030 0.84 CTSL (0.59) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7400378 0.83 CTSL (0.70) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7400382 0.83 CTSL (0.70) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7400374 0.83 CTSL (0.70) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7399923 0.81 CTSL (0.49) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7400387 0.81 CTSL (0.38) CTSLCTSBCTSSCTSKCTSH
SCHEMBL8516640 0.79 CTSL (0.64) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7411045 0.77 ACACB (0.46) CTSLCTSBCTSSMASP2F2
SCHEMBL7595864 0.75 CTSB (0.49) CTSLCTSBCTSSCTSKCTSH
SCHEMBL7414219 0.75 CTSB (0.49) CTSLCTSBCTSSCTSKCTSH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995023222-A1 IRREVERSIBLE CYSTEINE PROTEASE INHIBITORS CONTAINING VINYL GROUPS CONJUGATED TO ELECTRON WITHDRAWING GROUPS KHEPRI PHARMACEUTICALS, INC. (US) 1995-08-31 WO claimed