SCHEMBL7400423

SCHEMBL7400423

CCOC(=O)[C@H](Cc1ccc(CBr)cc1)N=C(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
AAK1 Q2M2I8 1/20 0.43
NPC1 O15118 1/20 0.43
MMP8 P22894 1/20 0.42
PPARG P37231 5/20 0.41
EPHX2 P34913 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PPARA Q07869 4/20 0.38
PIN1 Q13526 1/20 0.38
TP53 P04637 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151578 1.00 CES2 (0.44) CES2CES1MEN1KMT2AAAK1
SCHEMBL28584476 0.88 PPARG (0.45) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL5149030 0.86 ACHE (0.42) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL5310601 0.85 AAK1 (0.46) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL27559407 0.85 MEN1 (0.43) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL5155521 0.84 RORC (0.40) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL7222441 0.84 PPARG (0.43) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL5311248 0.84 AAK1 (0.42) CES2CES1MEN1KMT2AAAK1
SCHEMBL5155457 0.83 ACHE (0.43) MEN1KMT2AAAK1NPC1MMP8
SCHEMBL18554062 0.83 AAK1 (0.40) MEN1KMT2AAAK1NPC1MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690847-A1 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1996-01-10 EP disclosed
WO-1994022835-A2 HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS ZENECA LIMITED (GB) 1994-10-13 WO disclosed