SCHEMBL7400564

SCHEMBL7400564

Cc1cc(COc2ccc(C(=O)NC(C)C3(C(=O)NO)CCN(C(=O)OC(C)(C)C)CC3)cc2)c2ccccc2n1

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 11/20 0.70
MMP2 P08253 2/20 0.68
MMP13 P45452 2/20 0.68
MMP12 P39900 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595325 0.85 ADAM17 (0.74) ADAM17MMP2MMP13MMP12
SCHEMBL6596502 0.85 ADAM17 (0.72) ADAM17MMP2MMP13MMP12
SCHEMBL7400898 0.85 ADAM17 (0.67) ADAM17MMP2MMP13MMP12
SCHEMBL7400562 0.84 ADAM17 (0.70) ADAM17MMP2MMP13MMP12
SCHEMBL6600428 0.82 ADAM17 (1.00) ADAM17MMP13
SCHEMBL6596322 0.80 ADAM17 (0.75) ADAM17MMP2MMP13
SCHEMBL5221455 0.80 ADAM17 (0.85) ADAM17MMP13
SCHEMBL6597920 0.80 ADAM17 (0.64) ADAM17MMP2MMP13MMP12
SCHEMBL7404746 0.78 ADAM17 (0.62) ADAM17MMP2MMP13MMP12
SCHEMBL6598627 0.78 ADAM17 (0.84) ADAM17MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263756-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA Bristol-Myers Squibb Pharma Company (US) 2002-12-11 EP disclosed
WO-2001070734-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-09-27 WO disclosed