SCHEMBL7400587

SCHEMBL7400587

COc1cc(-c2nc3cc(C)c(C)cc3[nH]2)ccc1O

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 9/20 0.65
GUSB P08236 3/20 0.60
CYP1A1 P04798 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP1B1 Q16678 1/20 0.57
ALOX5 P09917 1/20 0.56
EPHX2 P34913 1/20 0.56
NOX1 Q9Y5S8 2/20 0.56
CHEK1 O14757 1/20 0.54
PARP1 P09874 1/20 0.53
HPSE Q9Y251 1/20 0.52
MGAM O43451 1/20 0.52
GAA P10253 1/20 0.52
SI P14410 1/20 0.52
MGAM2 Q2M2H8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7396876 0.85 ALOX5 (0.62) AMY1AGUSBCYP1A1CYP1A2CYP1B1
SCHEMBL7396878 0.85 ALOX5 (0.78) AMY1ACYP1A1CYP1A2CYP1B1ALOX5
SCHEMBL15456540 0.82 CYP1A1 (0.69) AMY1AGUSBCYP1A1CYP1A2CYP1B1
SCHEMBL7395696 0.82 AMY1A (0.77) AMY1ACYP1A1CYP1A2CYP1B1ALOX5
SCHEMBL7395692 0.82 AMY1A (0.62) AMY1ACYP1A1CYP1A2CYP1B1ALOX5
SCHEMBL7271955 0.79 KDM4E (0.62) AMY1AGUSBCYP1A1CYP1A2CYP1B1
SCHEMBL31737379 0.79 CYP1A1 (0.58) GUSBCYP1A1CYP1A2CYP1B1NOX1
SCHEMBL15224066 0.79 CYP1A1 (0.55) AMY1ACYP1A1CYP1A2CYP1B1ALOX5
SCHEMBL12470812 0.79 CYP1A1 (0.58) GUSBCYP1A1CYP1A2CYP1B1NOX1
SCHEMBL7997763 0.79 CYP1A1 (0.52) AMY1AGUSBCYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001066526-A1 ESTER DERIVATIVES OF DIMETHYLPROPIONIC ACID AND PHARMACETUICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2001-09-13 WO disclosed
EP-1132381-A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them CERMOL S.A. (CH) 2001-09-12 EP disclosed