SCHEMBL7400753

SCHEMBL7400753

N#Cc1ccc([N+]2([O-])CCNC2)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.33
CYP2A6 P11509 2/20 0.33
CA12 O43570 2/20 0.33
CA9 Q16790 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA1 P00915 3/20 0.32
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
PNMT P11086 1/20 0.32
TSHR P16473 1/20 0.31
OPRD1 P41143 1/20 0.31
CHRNA10 Q9GZZ6 1/20 0.31
CHRNA9 Q9UGM1 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
MMP3 P08254 1/20 0.31
ENPP2 Q13822 1/20 0.31
CHRNA1 P02708 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15415315 0.79
SCHEMBL11678412 0.78 MEN1 (0.31)
SCHEMBL11880913 0.72 ALDH1A1 (0.42) CA2CA12CA9ALDH1A1CA3
SCHEMBL8672077 0.67 TRPV1 (0.32) ALDH1A1TSHR
Hydrochloric Acid SCHEMBL8646091 0.67 HRH2 (0.35) CA2CA12CA9CA1LOXL2
SCHEMBL8580198 0.67 HTT (0.36) ALDH1A1TSHR
SCHEMBL3781336 0.66 CHRNB2 (0.36) CYP2A6ALDH1A1CHRNB2CHRNA4
SCHEMBL10741029 0.66 HTR2C (0.37) ALDH1A1TSHR
SCHEMBL5392162 0.65 ORAI1 (0.38) TSHR
SCHEMBL45942 0.63 CA2 (0.69) CA2CYP2A6CA12CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715623-B1 PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1998-09-09 EP disclosed
EP-0715623-A1 PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1996-06-12 EP disclosed
US-5489594-A ANTICOAGULANTS G. D. SEARLE & CO. (US) 1996-02-06 US disclosed
US-5430043-A Platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-07-04 US disclosed
WO-1995006038-A1 PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1995-03-02 WO disclosed