SCHEMBL7400768

SCHEMBL7400768

Cc1ccc2c(c1)nc(Cl)c1cccn12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 4/20 0.57
HTR3B O95264 4/20 0.57
HTR3A P46098 4/20 0.57
HTR3D Q70Z44 4/20 0.57
HTR3C Q8WXA8 4/20 0.57
PTPN1 P18031 3/20 0.53
HTR1A P08908 1/20 0.49
PTPN2 P17706 1/20 0.47
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HTT P42858 2/20 0.44
HPGD P15428 1/20 0.44
PDE10A Q9Y233 1/20 0.42
RAD51 Q06609 4/20 0.42
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NLRP3 Q96P20 1/20 0.40
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401133 0.83 PTPN1 (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1079670 0.81 RAD51 (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL13082235 0.81 RAD51 (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1309484 0.81 RAD51 (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7400933 0.80 RAD51 (0.61) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8569855 0.79 PTPN1 (0.61) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL27077503 0.78 PTPN1 (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL3789425 0.77 KDM4E (0.61) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL29893072 0.75 KDM4E (0.50) PTPN1KDM4EHTTRAD51MAPT
SCHEMBL24553486 0.73 ALDH1A1 (0.60) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001014381-A1 ETHER DERIVATIVES OF PYRROLO[1,2-A]QUINOXALINES, METHOD FOR PRODUCING THEM AND THEIR USE IN THERAPY UNIVERSITE DE CAEN BASSE-NORMANDIE (FR) 2001-03-01 WO disclosed
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed