SCHEMBL7400933

SCHEMBL7400933

COc1ccc2c(c1)nc(Cl)c1cccn12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD51 Q06609 5/20 0.61
HTR1A P08908 2/20 0.52
HTR3E A5X5Y0 1/20 0.52
HTR3B O95264 1/20 0.52
HTR3A P46098 1/20 0.52
HTR3D Q70Z44 1/20 0.52
HTR3C Q8WXA8 1/20 0.52
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 4/20 0.51
HPGD P15428 2/20 0.51
MAPT P10636 1/20 0.51
HTR2C P28335 1/20 0.47
PTPN1 P18031 1/20 0.46
POLB P06746 2/20 0.45
HTT P42858 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
TDP1 Q9NUW8 1/20 0.44
GFER P55789 1/20 0.44
NPC1 O15118 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400768 0.80 HTR3E (0.57) RAD51HTR1AHTR3EHTR3BHTR3A
SCHEMBL7401133 0.80 PTPN1 (0.54) RAD51HTR1AHTR3EHTR3BHTR3A
SCHEMBL18584266 0.77 RAD51 (0.44) RAD51HTR1AHTR3EHTR3BHTR3A
SCHEMBL1079670 0.77 RAD51 (0.58) RAD51HTR1AHTR3EHTR3BHTR3A
SCHEMBL13082235 0.77 RAD51 (0.51) RAD51HTR3EHTR3BHTR3AHTR3D
SCHEMBL29893072 0.77 KDM4E (0.50) RAD51KDM4EMAPTPTPN1HTT
SCHEMBL20816322 0.76 RAD51 (1.00) RAD51ALDH1A1KDM4EHPGDMAPT
SCHEMBL20816301 0.76 RAD51 (1.00) RAD51ALDH1A1KDM4EHPGDMAPT
SCHEMBL8569855 0.76 PTPN1 (0.61) RAD51HTR1AHTR3EHTR3BHTR3A
SCHEMBL8570795 0.75 HTR3E (0.72) HTR1AHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001014381-A1 ETHER DERIVATIVES OF PYRROLO[1,2-A]QUINOXALINES, METHOD FOR PRODUCING THEM AND THEIR USE IN THERAPY UNIVERSITE DE CAEN BASSE-NORMANDIE (FR) 2001-03-01 WO disclosed
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed