SCHEMBL7401316

SCHEMBL7401316

O=C(C#CCO)NCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.49
MCL1 Q07820 1/20 0.49
ALDH1A1 P00352 4/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 2/20 0.47
EPHX2 P34913 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RIPK1 Q13546 1/20 0.47
KMT2A Q03164 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 2/20 0.47
TSHR P16473 2/20 0.47
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
PADI3 Q9ULW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394877 0.84 MCL1 (0.47) GAAMCL1ALDH1A1LMNAHPGD
SCHEMBL31427583 0.84 RIPK1 (0.54) GAAMCL1ALDH1A1EPHX2L3MBTL1
SCHEMBL28350981 0.79 NPC1 (0.49) GAAMCL1ALDH1A1HPGDEPHX2
SCHEMBL5527107 0.77 GAA (0.55) GAAMCL1ALDH1A1LMNAHPGD
SCHEMBL14336905 0.76 ALDH1A1 (0.49) GAAMCL1ALDH1A1HPGDEPHX2
SCHEMBL669951 0.76 GAA (0.53) GAAMCL1ALDH1A1LMNAHPGD
SCHEMBL653442 0.76 MCL1 (0.62) GAAMCL1ALDH1A1LMNAHPGD
SCHEMBL21847278 0.72 L3MBTL1 (0.59) GAAMCL1ALDH1A1LMNAHPGD
SCHEMBL714625 0.72 EPHX1 (0.77) GAAALDH1A1LMNAHPGDEPHX2
SCHEMBL3056874 0.72 KMT2A (0.71) GAAALDH1A1LMNAHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711162-A4 IMIDAZOLE 5-POSITION SUBSTITUTED ANGIOTENSIN II ANTAGONISTS DU PONT MERCK PHARMA (US) 1996-09-04 EP disclosed
US-5545651-A HYPOTENSIVE AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1996-08-13 US disclosed
EP-0711162-A1 IMIDAZOLE 5-POSITION SUBSTITUTED ANGIOTENSIN II ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-05-15 EP disclosed
US-5395844-A Hypotensive agents; congestive heart failure THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-03-07 US disclosed
WO-1994028896-A1 IMIDAZOLE 5-POSITION SUBSTITUTED ANGIOTENSIN II ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-12-22 WO disclosed