SCHEMBL7401410

SCHEMBL7401410

CCCC(NC(=O)C(CC(C)C)c1ccc(-c2ccc(N3CCN(C4CCNCC4)CC3)cc2)cc1)C(=O)c1nc2ccccc2o1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.43
CTSK P43235 8/20 0.43
CTSL P07711 7/20 0.43
CTSB P07858 7/20 0.43
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7398214 0.92 CTSS (0.47) CTSSCTSKCTSLCTSBCYP3A4
SCHEMBL7444842 0.86 CTSK (0.56) CTSSCTSKCTSLCTSB
SCHEMBL7437343 0.79 CTSS (0.38) CTSSCTSKCTSLCTSBCYP3A4
SCHEMBL7402887 0.73 CTSS (0.47) CTSSCTSKCTSLCTSBCYP2C9
SCHEMBL7401526 0.73 CTSS (0.47) CTSSCYP3A4CYP2C9
SCHEMBL7402990 0.69 CTSS (0.45) CTSSCYP3A4CYP2C9
SCHEMBL7400014 0.69 CTSK (0.61) CTSSCTSKCTSLCTSB
SCHEMBL7048560 0.68 CTSS (0.82) CTSSCTSKCTSLCTSBCYP3A4
SCHEMBL6062148 0.67 CTSS (0.46) CTSSCTSKCTSLCTSBCYP3A4
SCHEMBL27663433 0.67 CTSS (0.50) CTSSCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002080920-A1 ARYLACETAMIDO-KETOBENZOXAZOLE AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-10-17 WO claimed